TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]WIN-35428 form human DAT expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 10.6nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 14.7nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 16.3nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in rat PC12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 37.1nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 49.7nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 53.8nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 96nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 101nMAssay Description:Displacement of [3H]WIN-35428 form human DAT expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 177nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 184nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 188nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 198nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in rat PC12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 198nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 232nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 232nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 244nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 259nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 262nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 302nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 373nMAssay Description:Binding affinity to 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 468nMAssay Description:Binding affinity to 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 469nMAssay Description:Binding affinity to 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 488nMAssay Description:Displacement of [3H]pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 497nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 599nMAssay Description:Binding affinity to 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 655nMAssay Description:Binding affinity to 5HT2BMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 705nMAssay Description:Inhibition of muscarinic M4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 774nMAssay Description:Binding affinity to 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 806nMAssay Description:Binding affinity to 5HT1AMore data for this Ligand-Target Pair