Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: <0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: <0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: <0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of rat Nav1.7 stably expressed in cells with train pulses to -20 mV at 0.1 Hz and holding potential of -90 mV by whole-cell QPatch HT assa...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human PAR-1 expressed in HEK293 cells assessed as reduction in TRAP induced calcium signal at 3 uM by FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human Nav1.7 stably expressed in cells with train pulses to -20 mV at 0.1 Hz and holding potential of -95 mV by whole-cell QPatch HT as...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human PAR-1 expressed in HEK293 cells assessed as reduction in TRAP induced calcium signal at 3 uM by FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human PAR-1 expressed in HEK293 cells assessed as reduction in TRAP induced calcium signal at 3 uM by FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of gamma secretase-mediated amyloid-beta peptid aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
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