TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:Binding affinity for mutant T877A Androgen receptor in human LNCaP cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 0.400nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity for mutant T877A Androgen receptor in human LNCaP cellsMore data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Inhibition of [3H]-DHT binding to T877A androgen receptor of LNCaP cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Inhibition of [3H]-DHT binding to T877A androgen receptor of LNCaP cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DHT from human androgen receptor in MDA453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of [3H]-DHT binding to androgen receptor of MDA-453 cellsMore data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-DHT from androgen receptor of human MDA-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 1.5nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair