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Found 362 with Last Name = 'dhanoa' and Initial = 'd'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187381(CHEMBL209324 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187394(CHEMBL207220 | N-(3-{4-[4-(cyclohexylmethanesulfon...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187377(CHEMBL209821 | N-(3-(4-(4-(cyclohexylmethylsulfona...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50005127(1,1-Dioxo-2-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-b...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187381(CHEMBL209324 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1 receptor in rat cerebral cortex cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187387(CHEMBL210537 | N-(3-(4-(4-(4-methylphenylsulfonami...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  8nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187389(CHEMBL377697 | cyclopropanecarboxylic acid {3-[4-(...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187379(CHEMBL379984 | N-(3-{4-[4-(2-methyl-propane-1-sulf...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187383(CHEMBL207478 | N-[3-(4-{4-[methyl-(2-methyl-propan...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187385(CHEMBL211012 | N-{3-[4-(1-Cyclohexylmethanesulfony...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50403914(CHEMBL2113711)
Affinity DataKi:  10nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114973(CHEMBL51542 | N-(4-{[(Naphthalen-2-ylmethyl)-amino...)
Affinity DataKi:  10nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114977(CHEMBL51884 | Naphthalene-1-sulfonic acid (4-{[(1,...)
Affinity DataKi:  11nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187381(CHEMBL209324 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]RX 821002 from Adrenergic alpha-2a receptor in rat cerebral cortex cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50005132(4,4-Dimethyl-1-[4-(4-pyrimidin-2-yl-piperazin-1-yl...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187376(CHEMBL210874 | N-(3-(4-((1-(4-fluorophenylsulfonyl...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50001859((buspirone) 8-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)...)
Affinity DataKi:  13nMAssay Description:Binding affinity to D2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114976(2-Nitro-N-(4-{[(quinolin-2-ylmethyl)-amino]-methyl...)
Affinity DataKi:  14nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114979(CHEMBL415926 | Naphthalene-2-sulfonic acid (4-{[(1...)
Affinity DataKi:  14nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114978(CHEMBL299295 | Naphthalene-1-sulfonic acid (4-{[2-...)
Affinity DataKi:  17nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187377(CHEMBL209821 | N-(3-(4-(4-(cyclohexylmethylsulfona...)
Affinity DataKi:  17nMAssay Description:Binding affinity to 5HT1A receptor in rat cerebral cortex by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Rat 6B)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  18nMAssay Description:Functional response of NPY to inhibit forskolin-stimulated cAMP in cells stably transfected with rat Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187393(CHEMBL210795 | N-(3-{4-[4-(4-fluoro-benzenesulfony...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403726(CHEMBL2112936)
Affinity DataKi:  20nMAssay Description:Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 2 betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50001859((buspirone) 8-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187378(CHEMBL209459 | cyclopropanecarboxylic acid (3-{4-[...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187388(CHEMBL209985 | N-(3-{4-[4-(propane-2-sulfonylamino...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114981(CHEMBL51874 | N-(4-{[(Naphthalen-1-ylmethyl)-amino...)
Affinity DataKi:  26nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114980(2-Nitro-N-(4-{[(quinolin-4-ylmethyl)-amino]-methyl...)
Affinity DataKi:  28nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187381(CHEMBL209324 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  30nMAssay Description:Binding affinity to 5HT7 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187390(CHEMBL380369 | Sunepitron)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1 receptor in rat cerebral cortex cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187397(CHEMBL266832 | N-(3-(4-(4-(cyclohexylsulfonylamino...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187380(4-methyl-N-(4-(4-phenylpiperazin-1-yl)butyl)benzen...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50075917(8N-(2-aminoethyl)-15-oxo-9a,10,11,12,13,13a,14,15-...)
Affinity DataKi:  45nMAssay Description:Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 2 betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187395(CHEMBL205550 | N-{4-[4-(3-methanesulfonylamino-phe...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187396(4-methyl-N-(4-{4-[3-(propane-2-sulfonylamino)-phen...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187381(CHEMBL209324 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  53nMAssay Description:Binding affinity to 5HT2B receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187398(CHEMBL445928 | N-(3-{4-[4-(toluene-4-sulfonylamino...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50005132(4,4-Dimethyl-1-[4-(4-pyrimidin-2-yl-piperazin-1-yl...)
Affinity DataKi:  58nMAssay Description:Binding affinity to D2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  63nMAssay Description:Binding affinity of the compound against cloned human Dopamine receptor D2 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403725(CHEMBL2112326)
Affinity DataKi:  75nMAssay Description:Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 2 betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187391(CHEMBL379364 | N-(3-{4-[4-(toluene-4-sulfonylamino...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50075918(8N-[2-amino-(1R,2R)-cyclohexyl]-15-oxo-(9aS,13aS)-...)
Affinity DataKi:  86nMAssay Description:Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 2 betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187390(CHEMBL380369 | Sunepitron)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  100nMAssay Description:Bnding affinity of the compound against cloned human Alpha-2C adrenergic receptor was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187377(CHEMBL209821 | N-(3-(4-(4-(cyclohexylmethylsulfona...)
Affinity DataKi:  100nMAssay Description:Binding affinity to guinea pig sigma receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50005127(1,1-Dioxo-2-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-b...)
Affinity DataKi:  110nMAssay Description:Binding affinity to D2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403726(CHEMBL2112936)
Affinity DataKi:  110nMAssay Description:Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Predix Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50187386(CHEMBL384677 | N-(3-{4-[1-(propane-2-sulfonyl)-pip...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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