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Found 47 with Last Name = 'salehian' and Initial = 'f'
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059510(8-Methoxy-3-phenyl-1,2,3,4-tetrahydro-chromeno[3,4...)
Affinity DataKi:  0nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059503(8-Methoxy-3-pyridin-4-ylmethyl-1,2,3,4-tetrahydro-...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to D4 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059507(3-Benzyl-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059505(3-(4-Chloro-benzyl)-8-hydroxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059504(8-Methoxy-3-(4-methyl-benzyl)-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059496(3-Benzyl-8-methyl-1,2,3,4-tetrahydro-chromeno[3,4-...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059491(3-(4-Fluoro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059492(3-(4-Fluoro-benzyl)-8-methyl-1,2,3,4-tetrahydro-ch...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059497(8-Methoxy-3-phenethyl-1,2,3,4-tetrahydro-chromeno[...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059501(8-Methoxy-3-(4-trifluoromethyl-benzyl)-1,2,3,4-tet...)
Affinity DataKi:  8.20nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059493(3-(4-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  8.70nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059499(3-(4-Chloro-benzyl)-8-methyl-1,2,3,4-tetrahydro-ch...)
Affinity DataKi:  11nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059494(3-(3-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  17nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059511(3-(2-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  34nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059507(3-Benzyl-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4...)
Affinity DataKi:  60nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059498(3-(3,4-Dichloro-benzyl)-8-methoxy-1,2,3,4-tetrahyd...)
Affinity DataKi:  61nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059503(8-Methoxy-3-pyridin-4-ylmethyl-1,2,3,4-tetrahydro-...)
Affinity DataKi:  74nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059502(8-Methoxy-3-(4-methoxy-benzyl)-1,2,3,4-tetrahydro-...)
Affinity DataKi:  84nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059505(3-(4-Chloro-benzyl)-8-hydroxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  317nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059496(3-Benzyl-8-methyl-1,2,3,4-tetrahydro-chromeno[3,4-...)
Affinity DataKi:  338nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059507(3-Benzyl-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4...)
Affinity DataKi:  436nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059504(8-Methoxy-3-(4-methyl-benzyl)-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  491nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059491(3-(4-Fluoro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  548nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059497(8-Methoxy-3-phenethyl-1,2,3,4-tetrahydro-chromeno[...)
Affinity DataKi:  591nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059496(3-Benzyl-8-methyl-1,2,3,4-tetrahydro-chromeno[3,4-...)
Affinity DataKi:  774nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059501(8-Methoxy-3-(4-trifluoromethyl-benzyl)-1,2,3,4-tet...)
Affinity DataKi:  966nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059499(3-(4-Chloro-benzyl)-8-methyl-1,2,3,4-tetrahydro-ch...)
Affinity DataKi:  1.17E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059504(8-Methoxy-3-(4-methyl-benzyl)-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  1.17E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059492(3-(4-Fluoro-benzyl)-8-methyl-1,2,3,4-tetrahydro-ch...)
Affinity DataKi:  2.21E+3nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059511(3-(2-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  2.62E+3nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059494(3-(3-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  2.63E+3nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059505(3-(4-Chloro-benzyl)-8-hydroxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  2.78E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50059493(3-(4-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  2.78E+3nMAssay Description:Binding affinity to human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059510(8-Methoxy-3-phenyl-1,2,3,4-tetrahydro-chromeno[3,4...)
Affinity DataKi: >3.30E+3nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059501(8-Methoxy-3-(4-trifluoromethyl-benzyl)-1,2,3,4-tet...)
Affinity DataKi:  3.70E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059494(3-(3-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi:  5.50E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059511(3-(2-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi: >5.80E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059491(3-(4-Fluoro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi: >5.80E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059493(3-(4-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-c...)
Affinity DataKi: >5.80E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059498(3-(3,4-Dichloro-benzyl)-8-methoxy-1,2,3,4-tetrahyd...)
Affinity DataKi: >5.80E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059503(8-Methoxy-3-pyridin-4-ylmethyl-1,2,3,4-tetrahydro-...)
Affinity DataKi: >5.80E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059497(8-Methoxy-3-phenethyl-1,2,3,4-tetrahydro-chromeno[...)
Affinity DataKi: >5.80E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059492(3-(4-Fluoro-benzyl)-8-methyl-1,2,3,4-tetrahydro-ch...)
Affinity DataKi: >5.80E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50059502(8-Methoxy-3-(4-methoxy-benzyl)-1,2,3,4-tetrahydro-...)
Affinity DataKi: >5.80E+3nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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LigandPNGBDBM50363804(CHEMBL1946917)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
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TargetDNA topoisomerase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50363804(CHEMBL1946917)
Affinity DataIC50:  39nMAssay Description:Inhibition of DNA topoisomerase 1 (unknown origin) at 50 uM measured by agar gel electrophoresisMore data for this Ligand-Target Pair
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LigandPNGBDBM50363797(CHEMBL1947110)
Affinity DataIC50:  67nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
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