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TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM50070214(4-(7,7-Dimethyl-oct-3-ynyl)-1H-imidazole | CHEMBL2...)
Affinity DataKi:  0.830nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM50070220(4-(6-Cyclopentyl-hex-3-ynyl)-1H-imidazole | CHEMBL...)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85407(GT 2231)
In DepthDetails PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM50070211(4-(6-Cyclohexyl-hex-3-ynyl)-1H-imidazole | CHEMBL1...)
Affinity DataKi:  2.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Human)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85405(GT 2227 | GT 2228)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85412(GT 2287)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85405(GT 2227 | GT 2228)
Affinity DataKi:  4.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85402(GT 2327)
Affinity DataKi:  5.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319488(CHEMBL1084901 | rac-{5-Chloro-3-[2-(3,5-dimethyl-i...)
Affinity DataKi:  8nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85399(GT 2148)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319486(CHEMBL1084893 | rac-{3-[2-(3,5-Dimethyl-isoxazol-4...)
Affinity DataKi:  12nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162903(CHEMBL359855 | [6-(4-Fluoro-benzenesulfonylamino)-...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319487(CHEMBL1084894 | rac-{2-Methyl-3-[2-(3-methyl-5-phe...)
Affinity DataKi:  13nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85405(GT 2227 | GT 2228)
Affinity DataKi:  15.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85411(GT 2174)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319482(CHEMBL1082939 | rac-{3-[2-(3,5-Dimethyl-isoxazol-4...)
Affinity DataKi:  18nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)
Affinity DataKi:  18nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 in hTP binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162894(CHEMBL361972 | [2-(4-Fluoro-benzenesulfonylamino)-...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319495(CHEMBL1082610 | rac-{3-[2-(3,5-Dimethyl-isoxazol-4...)
Affinity DataKi:  23nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319486(CHEMBL1084893 | rac-{3-[2-(3,5-Dimethyl-isoxazol-4...)
Affinity DataKi:  28nMAssay Description:Antagonist activity at human prostaglandin D2 receptor assessed as inhibition of PGD2-induced receptor activation by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319490(CHEMBL1084903 | rac-{3-[1,1-Dioxo-2-(2-phenoxy-eth...)
Affinity DataKi:  29nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162917(CHEMBL360288 | [6-(4-Fluoro-benzenesulfonylamino)-...)
Affinity DataKi:  30nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85401(GT 2140)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319491(CHEMBL1083446 | rac-(3-{2-[2-(4-Chloro-phenoxy)-et...)
Affinity DataKi:  35nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319494(CHEMBL1085069 | rac-{3-[2-(3,5-Dimethyl-isoxazol-4...)
Affinity DataKi:  38nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162891(CHEMBL179980 | [6-(4-Fluoro-benzenesulfonylamino)-...)
Affinity DataKi:  50nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85406(GT 2321)
Affinity DataKi:  75nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85403(GT 2130)
Affinity DataKi:  104nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162896(CHEMBL369330 | [3-tert-Butyl-6-(4-fluoro-benzenesu...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162901(CHEMBL180733 | [5-(4-Fluoro-benzenesulfonylamino)-...)
Affinity DataKi:  200nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319489(CHEMBL1084902 | rac-[3-(1,1-Dioxo-2-phenethyl-2,3-...)
Affinity DataKi:  220nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162897(3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)
Affinity DataKi:  250nMAssay Description:Inhibitory activity of the compound against CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162897(3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)
Affinity DataKi:  250nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)
Affinity DataKi:  290nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)
Affinity DataKi:  290nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)
Affinity DataKi:  340nMAssay Description:Inhibitory concentration of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319477(CHEMBL1086341 | rac-[3-(1,1-Dioxo-2,3-dihydro-1H-1...)
Affinity DataKi:  430nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319485(CHEMBL1085645 | rac-[3-(1,1-Dioxo-2-phenyl-2,3-dih...)
Affinity DataKi:  480nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319483(CHEMBL1085640 | rac-{2-Methyl-3-[2-(3-methyl-butyl...)
Affinity DataKi:  560nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319481(CHEMBL1085639 | rac-[3-(1,1-Dioxo-2-phenethyl-2,3-...)
Affinity DataKi:  630nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85404(GT 2146)
Affinity DataKi:  630nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319476(CHEMBL1083158 | rac-[5-Chloro-3-(1,1-dioxo-2,3-dih...)
Affinity DataKi:  690nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319484(CHEMBL1085644 | rac-[3-(2-Isopropyl-1,1-dioxo-2,3-...)
Affinity DataKi:  920nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162925(3-[6-(2-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)
Affinity DataKi:  970nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM85408(GT 2288)
Affinity DataKi:  1.03E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319480(CHEMBL1086343 | rac-[3-(2-Benzyl-1,1-dioxo-2,3-dih...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162902(3-(6-Benzenesulfonylamino-1,2,3,4-tetrahydro-carba...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50162892(3-[6-(3-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Human)
Athersys

Curated by ChEMBL
LigandPNGBDBM50319492(CHEMBL1083752 | rac-{3-[1,1-Dioxo-2-(3-phenoxy-pro...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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