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Found 192 with Last Name = 'heitsch' and Initial = 'h'
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50075000((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074978(2-[3-(4-Amino-butyl)-ureido]-N-[4-chloro-2-cyano-3...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074986((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074997((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[4-methoxy-...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074993((E)-N-({[2,4-Dimethyl-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074982((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074983((E)-N-({[2-Chloro-4-methoxy-3-(2-methyl-quinolin-8...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074984((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074992((E)-N-({[4-Chloro-2-methoxy-3-(2-methyl-quinolin-8...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074980((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074990(4-[3-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-yl...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074991((E)-Penta-2,4-dienoic acid ({[2,4-dichloro-3-(2-me...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074985((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074998((E)-N-({[4-Methoxy-3-(2-methyl-quinolin-8-yloxymet...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074994(5-[({[4-Methoxy-3-(2-methyl-quinolin-8-yloxymethyl...)
Affinity DataKi:  5.40nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074987(CHEMBL113502 | N-[2-Cyano-4-methoxy-3-(2-methyl-qu...)
Affinity DataKi:  6nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074979((E)-3-(4-Methoxy-phenyl)-N-({methyl-[3-(2-methyl-q...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074999(CHEMBL114180 | N-[4-Chloro-2-cyano-3-(2-methyl-qui...)
Affinity DataKi:  8.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074996(({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-yloxyme...)
Affinity DataKi:  9.10nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074981((E)-N-({[2,4-Dimethoxy-3-(2-methyl-quinolin-8-ylox...)
Affinity DataKi:  9.20nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074995((E)-N-({[2-Methoxy-3-(2-methyl-quinolin-8-yloxymet...)
Affinity DataKi:  45nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074988((E)-N-({[3-(Benzothiazol-4-yloxymethyl)-2,4-dichlo...)
Affinity DataKi:  160nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074989((E)-N-({[2,4-Dichloro-3-(2-phenyl-benzothiazol-4-y...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470233(CHEMBL80177)
Affinity DataIC50:  0.0800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470229(CHEMBL76870)
Affinity DataIC50:  0.0900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470239(CHEMBL311312)
Affinity DataIC50:  0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470236(CHEMBL309313)
Affinity DataIC50:  0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045686(4-(4-Amino-piperidin-1-yl)-N-[1-(1-cyclohexylmethy...)
Affinity DataIC50:  0.130nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045691(CHEMBL94827 | Methyl-{2-[methyl-(morpholine-4-carb...)
Affinity DataIC50:  0.160nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045691(CHEMBL94827 | Methyl-{2-[methyl-(morpholine-4-carb...)
Affinity DataIC50:  0.160nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045687(2-Benzyl-N-[1-(1-cyclohexylmethyl-2,3-dihydroxy-5-...)
Affinity DataIC50:  0.170nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470250(CHEMBL77308)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50213569(CHEMBL78866)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470225(CHEMBL80700)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470226(CHEMBL311827)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470235(CHEMBL308135)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470206(CHEMBL445365)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50213557(CHEMBL309602)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50031491(2-propyl-4-(methythio)-1-[[[2'-[(propylamino)carbo...)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045683(4-(4-Amino-piperidin-1-yl)-2-benzyl-N-[1-(1-cycloh...)
Affinity DataIC50:  0.240nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045685(4-(4-Amino-piperidin-1-yl)-2-benzyl-N-[1-(1-cycloh...)
Affinity DataIC50:  0.25nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045685(4-(4-Amino-piperidin-1-yl)-2-benzyl-N-[1-(1-cycloh...)
Affinity DataIC50:  0.260nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470249(CHEMBL309845)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470241(CHEMBL305638)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50031537(2-Butyl-3-(N'-propylureidylsulfonyl-biphenyl-4-ylm...)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470227(CHEMBL76538)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470223(CHEMBL312386)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045692(3-(4-Amino-cyclohexanesulfonyl)-2-benzyl-N-[1-(1-c...)
Affinity DataIC50:  0.310nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045692(3-(4-Amino-cyclohexanesulfonyl)-2-benzyl-N-[1-(1-c...)
Affinity DataIC50:  0.310nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045693(4-Amino-piperidine-1-carboxylic acid 1-[1-(1-cyclo...)
Affinity DataIC50:  0.370nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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