Affinity DataKi: <3.16E+3nMAssay Description:Binding affinity to 5HT1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: <3.16E+3nMAssay Description:Binding affinity to 5HT1B receptorMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.21E+5nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.05E+5nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.23E+5nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: >9.58E+5nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: >1.10E+6nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.36E+6nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R.W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: >1.38E+6nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Activity of the compound against thromboxane A2 receptor evaluated by contraction of isolated rat thoracic aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 324nMAssay Description:Activity of the compound against thromboxane A2 receptor evaluated by contraction of isolated rat thoracic aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Activity of the compound against thromboxane A2 receptor evaluated by aggregation of human plateletsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.11E+3nMAssay Description:Activity of the compound against thromboxane A2 receptor evaluated by aggregation of human plateletsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Activity of the compound against thromboxane A2 receptor evaluated by contraction of isolated rat thoracic aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 58nMAssay Description:Activity of the compound against thromboxane A2 receptor evaluated by contraction of isolated rat thoracic aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Transcriptional activation for RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Transcriptional activation for RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 275nMAssay Description:Transcriptional activation for RXR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4.58E+3nMAssay Description:Transcriptional activation for RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.5nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Transcriptional activation for RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 91nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 298nMAssay Description:Transcriptional activation for RXR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 74nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 77nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 152nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Transcriptional activation for RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 989nMAssay Description:Transcriptional activation for RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Transcriptional activation for RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.5nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 385nMAssay Description:Transcriptional activation for RXR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 195nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Transcriptional activation for RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.22E+3nMAssay Description:Transcriptional activation for RXR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Transcriptional activation for RXR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 961nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 102nMAssay Description:Transcriptional activation for RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: >6.40E+3nMAssay Description:Transcriptional activation for RXR alpha receptorMore data for this Ligand-Target Pair