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Found 196 with Last Name = 'sakai' and Initial = 'h'
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198670(CHEMBL3960590)
Affinity DataIC50:  24nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198661(CHEMBL3955849)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198660(CHEMBL3928231)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198677(CHEMBL3929427)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50460879(CHEMBL4228441)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant human KLK7 using MOCAc-Arg-Pro-Lys-Pro-Val-Glu-Nva-Trp-Arg-Lys(Dnp)-NH2 as substrate preincubated for 10 mins followed by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198662(CHEMBL3966957)
Affinity DataIC50:  56nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50275974(CHEMBL4126936)
Affinity DataIC50:  58nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged KLK7 (E23 to H252 residues) using MOCAcArg-Pro-Lys-Pro-Val-Glu-Nva-Trp-Arg-Lys(Dnp)-NH2 as su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50275974(CHEMBL4126936)
Affinity DataIC50:  58nMAssay Description:Inhibition of recombinant human KLK7 using MOCAc-Arg-Pro-Lys-Pro-Val-Glu-Nva-Trp-Arg-Lys(Dnp)-NH2 as substrate preincubated for 10 mins followed by s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355243(CHEMBL1835836)
Affinity DataIC50:  65nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287288((S)-2-{(S)-2-[4-(4-Carbamimidoyl-phenoxy)-butyryla...)
Affinity DataIC50:  76nMAssay Description:Inhibition of ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50092111((S)-2-{(S)-2-[4-(4-Carbamimidoyl-phenoxy)-butyryla...)
Affinity DataIC50:  88nMAssay Description:Inhibition of human platelet adhesion to fibrinogenMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50092111((S)-2-{(S)-2-[4-(4-Carbamimidoyl-phenoxy)-butyryla...)
Affinity DataIC50:  100nMAssay Description:Inhibition of ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKallikrein-7(Homo sapiens (Human))
Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50460884(CHEMBL4228178)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant human KLK7 using MOCAc-Arg-Pro-Lys-Pro-Val-Glu-Nva-Trp-Arg-Lys(Dnp)-NH2 as substrate preincubated for 10 mins followed by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287287((S)-3-[4-(4-Carbamimidoyl-phenoxy)-butyrylamino]-N...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [125I]- Fg binding to fibrinogen receptor of activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198682(CHEMBL3918835)
Affinity DataIC50:  120nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355241(CHEMBL1835834)
Affinity DataIC50:  120nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287286((S)-2-{(S)-2-[4-(4-Carbamimidoyl-phenoxy)-butyryla...)
Affinity DataIC50:  130nMAssay Description:Inhibition of ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50421378(CHEMBL146281)
Affinity DataIC50:  140nMAssay Description:Inhibition of ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198678(CHEMBL3891045)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198667(CHEMBL3963507)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198681(CHEMBL3966515)
Affinity DataIC50:  150nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198680(CHEMBL3983437)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198660(CHEMBL3928231)
Affinity DataIC50:  160nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from recombinant human GST-tagged PR-LBD (675 to 933 residues) expressed in baculovirus-infected insect cell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287282((S)-3-[4-(4-Carbamimidoyl-phenoxy)-butyrylamino]-N...)
Affinity DataIC50:  160nMAssay Description:Inhibition of ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198675(CHEMBL3957000)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355237(CHEMBL1835830)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198674(CHEMBL3965979)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198664(CHEMBL3954803)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355234(CHEMBL1835827)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355239(CHEMBL1835832)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198657(CHEMBL3960113)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198655(CHEMBL3948334)
Affinity DataIC50:  230nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287279((S)-2-{(S)-2-[5-(4-Carbamimidoyl-phenoxy)-pentanoy...)
Affinity DataIC50:  230nMAssay Description:Inhibition of ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366434(CHEMBL1790144)
Affinity DataIC50:  230nMAssay Description:Inhibition of ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287279((S)-2-{(S)-2-[5-(4-Carbamimidoyl-phenoxy)-pentanoy...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human platelet adhesion to fibrinogenMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198676(CHEMBL3936738)
Affinity DataIC50:  230nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198668(CHEMBL3955372)
Affinity DataIC50:  240nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198654(CHEMBL3927761)
Affinity DataIC50:  250nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355225(CHEMBL1835818)
Affinity DataIC50:  250nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355227(CHEMBL1835820)
Affinity DataIC50:  260nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198669(CHEMBL3938469)
Affinity DataIC50:  260nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287281((S)-3-[5-(4-Carbamimidoyl-phenoxy)-pentanoylamino]...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human platelet adhesion to fibrinogenMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287281((S)-3-[5-(4-Carbamimidoyl-phenoxy)-pentanoylamino]...)
Affinity DataIC50:  270nMAssay Description:Inhibition of ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198665(CHEMBL3894599)
Affinity DataIC50:  290nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355244(CHEMBL1835825)
Affinity DataIC50:  290nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198656(CHEMBL3946113)
Affinity DataIC50:  290nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198673(CHEMBL3975572)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355233(CHEMBL1835826)
Affinity DataIC50:  310nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198659(CHEMBL3946665)
Affinity DataIC50:  340nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355224(CHEMBL1835817)
Affinity DataIC50:  360nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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