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Found 240 with Last Name = 'ducharme' and Initial = 'j'
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120056(15-Amino-1-methyl-10-thia-tricyclo[7.5.1.0*2,7*]pe...)
Affinity DataKi:  0.790nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120057(7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetr...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120058(7-Amino-6-methoxy-8,8-dimethyl-5,6,7,8-tetrahydro-...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  4nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120053(7-Amino-6-ethyl-8,8-dimethyl-5,6,7,8-tetrahydro-na...)
Affinity DataKi:  21nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120056(15-Amino-1-methyl-10-thia-tricyclo[7.5.1.0*2,7*]pe...)
Affinity DataKi:  43nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  52nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120057(7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetr...)
Affinity DataKi:  66nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  113nMAssay Description:Binding affinity of the compound for Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120061(7-Amino-6-ethyl-8,8-dimethyl-5,6,7,8-tetrahydro-na...)
Affinity DataKi:  135nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120062(7-Amino-6-mercapto-8,8-dimethyl-5,6,7,8-tetrahydro...)
Affinity DataKi:  163nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120058(7-Amino-6-methoxy-8,8-dimethyl-5,6,7,8-tetrahydro-...)
Affinity DataKi:  184nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120054(3-Amino-4,4-dimethyl-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  204nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120059(7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetr...)
Affinity DataKi:  286nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120053(7-Amino-6-ethyl-8,8-dimethyl-5,6,7,8-tetrahydro-na...)
Affinity DataKi:  345nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120057(7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetr...)
Affinity DataKi:  349nMAssay Description:Binding affinity of the compound for Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120056(15-Amino-1-methyl-10-thia-tricyclo[7.5.1.0*2,7*]pe...)
Affinity DataKi:  420nMAssay Description:Binding affinity of the compound for Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120055(7-Amino-6-methanesulfinyl-8,8-dimethyl-5,6,7,8-tet...)
Affinity DataKi:  1.05E+3nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120055(7-Amino-6-methanesulfinyl-8,8-dimethyl-5,6,7,8-tet...)
Affinity DataKi:  1.06E+3nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120060(7-Amino-6-methanesulfonyl-8,8-dimethyl-5,6,7,8-tet...)
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120053(7-Amino-6-ethyl-8,8-dimethyl-5,6,7,8-tetrahydro-na...)
Affinity DataKi:  4.51E+3nMAssay Description:Binding affinity of the compound for Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120058(7-Amino-6-methoxy-8,8-dimethyl-5,6,7,8-tetrahydro-...)
Affinity DataKi:  5.22E+3nMAssay Description:Binding affinity of the compound for Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50039026(4-((R)-((2S,5R)-4-allyl-2,5-dimethylpiperazin-1-yl...)
Affinity DataIC50:  0.230nMAssay Description:Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092669(CHEMBL129420 | N,N-Diethyl-4-(piperazin-1-yl-quino...)
Affinity DataIC50:  0.510nMAssay Description:Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092704(CHEMBL339898 | N,N-Diethyl-4-[piperidin-4-ylidene-...)
Affinity DataIC50:  0.630nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092711(CHEMBL339457 | N,N-Diethyl-4-[(3-fluoro-phenyl)-pi...)
Affinity DataIC50:  0.740nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092703(4-[(3-Acetyl-phenyl)-piperidin-4-ylidene-methyl]-N...)
Affinity DataIC50:  0.860nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092710(CHEMBL415521 | N,N-Diethyl-4-(phenyl-piperidin-4-y...)
Affinity DataIC50:  0.870nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092701(CHEMBL278078 | N,N-Diethyl-4-[(2-methoxy-phenyl)-p...)
Affinity DataIC50:  0.970nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092712(CHEMBL126370 | N,N-Diethyl-4-[(2-fluoro-phenyl)-pi...)
Affinity DataIC50:  1nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092664(CHEMBL126819 | N,N-Diethyl-4-(piperazin-1-yl-quino...)
Affinity DataIC50:  1.10nMAssay Description:Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092716(CHEMBL340131 | N,N-Diethyl-4-[(3-nitro-phenyl)-pip...)
Affinity DataIC50:  1.10nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092676(4-[(2,2-Dimethyl-2,3-dihydro-benzofuran-7-yl)-pipe...)
Affinity DataIC50:  1.20nMAssay Description:Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092717(CHEMBL129034 | N,N-Diethyl-4-(naphthalen-1-yl-pipe...)
Affinity DataIC50:  1.20nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50039029((+)-4-((alpha R)-((2S,5R)-4-allyl-2,5-dimethylpipe...)
Affinity DataIC50:  1.30nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50039029((+)-4-((alpha R)-((2S,5R)-4-allyl-2,5-dimethylpipe...)
Affinity DataIC50:  1.30nMAssay Description:Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092706(CHEMBL423694 | N,N-Diethyl-4-[(3-methoxy-phenyl)-p...)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092715(CHEMBL339922 | N,N-Diethyl-4-[(4-methoxy-phenyl)-p...)
Affinity DataIC50:  2nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092702(CHEMBL129693 | N,N-Diethyl-4-[(4-methylsulfanyl-ph...)
Affinity DataIC50:  2.10nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092714(CHEMBL126141 | N,N-Diethyl-4-{[1-(3-methyl-but-2-e...)
Affinity DataIC50:  2.10nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50039026(4-((R)-((2S,5R)-4-allyl-2,5-dimethylpiperazin-1-yl...)
Affinity DataIC50:  2.10nMAssay Description:Binding affinity against cloned human Opioid receptor mu 1 using [125I]FK33824 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092719(4-[(3,4-Dichloro-phenyl)-piperidin-4-ylidene-methy...)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092680(CHEMBL125734 | N,N-Diethyl-4-(naphthalen-1-yl-pipe...)
Affinity DataIC50:  2.40nMAssay Description:Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092698(4-[(3-Amino-phenyl)-piperidin-4-ylidene-methyl]-N,...)
Affinity DataIC50:  2.60nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092720(CHEMBL129315 | N,N-Diethyl-4-(piperidin-4-ylidene-...)
Affinity DataIC50:  2.90nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092700(4-[(1-Allyl-piperidin-4-ylidene)-phenyl-methyl]-N,...)
Affinity DataIC50:  3nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092683(CHEMBL126366 | N,N-Diethyl-4-(isoquinolin-5-yl-pip...)
Affinity DataIC50:  4.10nMAssay Description:Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092709(4-[(4-Chloro-phenyl)-piperidin-4-ylidene-methyl]-N...)
Affinity DataIC50:  4.20nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092665(CHEMBL340834 | N,N-Diethyl-4-[(3-fluoro-phenyl)-pi...)
Affinity DataIC50:  4.5nMAssay Description:Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50092718(4-[(1-Butyl-piperidin-4-ylidene)-phenyl-methyl]-N,...)
Affinity DataIC50:  6.5nMAssay Description:Binding affinity on cloned opioid receptor delta 1 in human HEK293S cells using [125I]-[D-Ala2]-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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