Affinity DataKi: 0.300nMAssay Description:Binding affinity towards adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]CPX from rat brain cortex adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]CPX from rat brain cortex adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity towards adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX compared to SCH-58261 (Ki=390 nM)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]CPX from rat brain cortex adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H]CPX from rat brain cortex adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity towards adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX compared to SCH-58261 (Ki=390 nM)More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]CPX from rat brain cortex adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity towards adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX compared to SCH-58261 (Ki=390 nM)More data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity towards adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX compared to SCH-58261 (Ki=390 nM)More data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Tested in vitro for its inhibition of trifunctional glycinamide ribonucleotide formyltransferase (GARFT) isolated from murine L1210 leukemia cellsMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Displacement of [125I]3-(4-aminobenzyl)-8-phenyloxyacetate-1-propyl-xanthine from human adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 96nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [125I]3-(4-aminobenzyl)-8-phenyloxyacetate-1-propyl-xanthine from human adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 109nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity towards adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX compared to SCH-58261 (Ki=390 nM)More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity towards adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX compared to SCH-58261 (Ki=390 nM)More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Tested in vitro for its inhibition of trifunctional glycinamide ribonucleotide formyltransferase (GARFT) isolated from murine L1210 leukemia cellsMore data for this Ligand-Target Pair
Affinity DataKi: 127nMAssay Description:Displacement of [125I]3-(4-aminobenzyl)-8-phenyloxyacetate-1-propyl-xanthine from human adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Displacement of [125I]ZM241385 from human adenosine A2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair