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Found 122 with Last Name = 'gestwicki' and Initial = 'je'
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM50613636(CHEMBL5286207)
Affinity DataKi:  4nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM50613631(CHEMBL5281156)
Affinity DataKi:  6nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM50613624(CHEMBL5291300)
Affinity DataKi:  7nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM23334(3-(pyridin-3-yl)propyl (2S)-1-(3,3-dimethyl-2-oxop...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM50116636(1-(3,3-Dimethyl-2-oxo-pentanoyl)-pyrrolidine-2-car...)
Affinity DataKi:  11nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM50613623(CHEMBL5280097)
Affinity DataKi:  12nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM50132556((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataKi:  20nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM50613634(CHEMBL5289205)
Affinity DataKi:  23nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM50613635(CHEMBL5291024)
Affinity DataKi:  26nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM50030448(8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN | CHEMBL269732 ...)
Affinity DataKi:  93nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM912((3S,4S)-3-hydroxy-4-[(2S)-2-[(3S,4S)-3-hydroxy-6-m...)
Affinity DataKi:  94nMAssay Description:Inhibition of wild-type HIV-1 protease using fluorogenic peptide substrate incubated for 30 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM50067006((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataKi:  110nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM912((3S,4S)-3-hydroxy-4-[(2S)-2-[(3S,4S)-3-hydroxy-6-m...)
Affinity DataKi:  230nMAssay Description:Inhibition of multidrug resistant HIV-1 protease L10I/L63P/A71V/G73S/I84V/L90M mutant using fluorogenic peptide substrate incubated for 30 mins prior...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM50613625(CHEMBL1235853)
Affinity DataKi:  300nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM23334(3-(pyridin-3-yl)propyl (2S)-1-(3,3-dimethyl-2-oxop...)
Affinity DataKi:  306nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM23334(3-(pyridin-3-yl)propyl (2S)-1-(3,3-dimethyl-2-oxop...)
Affinity DataKi:  447nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM23334(3-(pyridin-3-yl)propyl (2S)-1-(3,3-dimethyl-2-oxop...)
Affinity DataKi:  936nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM50080534(CHEMBL333448 | ethyl (4-{(2R)-2-[(1S,3S,5S)-3,5-di...)
Affinity DataKi:  958nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM50080534(CHEMBL333448 | ethyl (4-{(2R)-2-[(1S,3S,5S)-3,5-di...)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))TBA
LigandPNGBDBM92915(Aryl 1-indanylketone, 4)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM50080534(CHEMBL333448 | ethyl (4-{(2R)-2-[(1S,3S,5S)-3,5-di...)
Affinity DataKi:  1.69E+3nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))TBA
LigandPNGBDBM50495808(CHEMBL1557710)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to CypD (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase B(Homo sapiens (Human))TBA
LigandPNGBDBM92915(Aryl 1-indanylketone, 4)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to CypB (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))TBA
LigandPNGBDBM50613627(CHEMBL2006156)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to CypD (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))TBA
LigandPNGBDBM50613626(CHEMBL5275318)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to CypD (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))TBA
LigandPNGBDBM50613626(CHEMBL5275318)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))TBA
LigandPNGBDBM50613627(CHEMBL2006156)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM50080528(3-((R)-2-((1S,3S,5S)-3,5-dimethyl-2-oxocyclohexyl)...)
Affinity DataKi:  3.40E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM50613621(CHEMBL5268083)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))TBA
LigandPNGBDBM50613621(CHEMBL5268083)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM50613621(CHEMBL5268083)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))TBA
LigandPNGBDBM50495808(CHEMBL1557710)
Affinity DataKi:  2.10E+4nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM50613633(CHEMBL5271713)
Affinity DataKi:  2.30E+4nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM50613635(CHEMBL5291024)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM50613636(CHEMBL5286207)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM50613634(CHEMBL5289205)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM50613631(CHEMBL5281156)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))TBA
LigandPNGBDBM50613632(CHEMBL5270994)
Affinity DataKi:  6.10E+4nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase B(Homo sapiens (Human))TBA
LigandPNGBDBM92920(Benzofuranone, 9)
Affinity DataKi:  6.30E+4nMAssay Description:Binding affinity to CypB (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50058936(CHEMBL3393116)
Affinity DataKi:  9.10E+4nMAssay Description:Inhibition of multidrug resistant HIV-1 protease L10I/L63P/A71V/G73S/I84V/L90M mutant using fluorogenic peptide substrate incubated for 30 mins prior...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50058936(CHEMBL3393116)
Affinity DataKi:  9.60E+4nMAssay Description:Inhibition of wild-type HIV-1 protease using fluorogenic peptide substrate incubated for 30 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM50613632(CHEMBL5270994)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))TBA
LigandPNGBDBM50613633(CHEMBL5271713)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))TBA
LigandPNGBDBM50613629(CHEMBL5268140)
Affinity DataIC50:  14nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50381013(CHEMBL2017129)
Affinity DataIC50:  200nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))TBA
LigandPNGBDBM50613628(CHEMBL5279925)
Affinity DataIC50:  300nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM34010(benzothiophene carboxamide, 18b)
Affinity DataIC50: <300nMAssay Description:Displacement of FITC-WFYpSPFLE from human Pin1 (45-163) catalytic domain by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))TBA
LigandPNGBDBM92913(Aryl 1-indanylketone, 2)
Affinity DataIC50:  300nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM92913(Aryl 1-indanylketone, 2)
Affinity DataIC50:  400nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))TBA
LigandPNGBDBM50381013(CHEMBL2017129)
Affinity DataIC50:  520nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
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