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Found 96 with Last Name = 'john' and Initial = 'jk'
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100510(3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-hexad...)
Affinity DataIC50:  130nMAssay Description:Inhibitory activity against P-selectin using ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100507(3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-hexad...)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity against P-selectin using ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50288934(2-[3,5-dihydroxy-2-(6-hydroxy-2-hydroxymethyl-4-ox...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against P-selectin using ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426811(US10544110, Compound MDV3100)
Affinity DataIC50:  1.10E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426809(US10544110, Compound JJ-450A)
Affinity DataIC50:  1.60E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426808(US10544110, Compound JJ-450)
Affinity DataIC50:  2.70E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100510(3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-hexad...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibitory activity against P-selectin using cell-selectin protein assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426799(US10544110, Compound 15)
Affinity DataIC50:  2.90E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100508(3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-dodec...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against P-selectin using ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426784(US10544110, Compound 5k)
Affinity DataIC50:  3.10E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426803(US10544110, Compound 18c)
Affinity DataIC50:  7.20E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM36974(2-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfanyl]-1...)
Affinity DataIC50:  7.30E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426806(US10544110, Compound 26a | US10544110, Compound 26...)
Affinity DataIC50:  7.70E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426806(US10544110, Compound 26a | US10544110, Compound 26...)
Affinity DataIC50:  7.90E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100510(3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-hexad...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against P-selectin using cell-cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100507(3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-hexad...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against P-selectin using cell-selectin protein assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426790(US10544110, Compound 6)
Affinity DataIC50:  1.08E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426779(US10544110, Compound 5g)
Affinity DataIC50:  1.11E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426783(US10544110, Compound 5j)
Affinity DataIC50:  1.11E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426777(US10544110, Compound 5e)
Affinity DataIC50:  1.20E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426778(US10544110, Compound 5f)
Affinity DataIC50:  1.26E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426798(US10544110, Compound 14)
Affinity DataIC50:  1.27E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426810(US10544110, Compound JJ-450B)
Affinity DataIC50:  1.31E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426791(US10544110, Compound 7)
Affinity DataIC50:  1.37E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100507(3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-hexad...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activity against P-selectin using cell-cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426792(US10544110, Compound 8)
Affinity DataIC50:  1.44E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426774(US10544110, Compound 5b)
Affinity DataIC50:  1.45E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426785(US10544110, Compound 5l)
Affinity DataIC50:  1.47E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100509(3-[4-(5-{4-[2-(4-Heptyl-phenylcarbamoyl)-vinyl]-ph...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory activity against P-selectin using ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426797(US10544110, Compound 13)
Affinity DataIC50:  1.61E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426786(US10544110, Compound 5m)
Affinity DataIC50:  1.66E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100506(3-(4-{5-[4-(2-Hexadecylcarbamoyl-vinyl)-phenyl]-1H...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory activity against P-selectin using ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426781(US10544110, Compound 5i)
Affinity DataIC50:  1.84E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100510(3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-hexad...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory activity against Selectin E using cell-cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426794(US10544110, Compound 10)
Affinity DataIC50:  2.03E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100511(3-[4-(2-[4-(2-Carboxy-vinyl)-phenyl]-5-{4-[2-(3-ph...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibitory activity against P-selectin using cell-selectin protein assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100514(3-(4-{5-[4-(2-Dihexylcarbamoyl-vinyl)-phenyl]-1H-i...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibitory activity against P-selectin using cell-selectin protein assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426773(US10544110, Compound 5a)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426775(US10544110, Compound 5c)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426776(US10544110, Compound 5d)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426780(US10544110, Compound 5h)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426793(US10544110, Compound 9)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426795(US10544110, Compound 11)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426796(US10544110, Compound 12)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426800(US10544110, Compound 16)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426801(US10544110, Compound 18a)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426802(US10544110, Compound 18b)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426804(US10544110, Compound 20a)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426805(US10544110, Compound 20b)
Affinity DataIC50: >2.50E+4nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE-selectin(Homo sapiens (Human))
Ontogen

Curated by ChEMBL
LigandPNGBDBM50100507(3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-hexad...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity against Selectin E using cell-cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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