TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0850nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Compound was evaluated for VCAM-VLA-4 antagonistic activity using solid phase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Cell Culture Conditions: CHO-K1 cells previously transfected with G-alpha 16 were subsequently transfected with the human CRTH2 receptor and the neom...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Very late antigen 4/vascular cell adhesion molecule 1 interaction in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of Very late antigen 4/vascular cell adhesion molecule 1 interaction in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibition of Very late antigen 4/vascular cell adhesion molecule 1 interaction in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Inhibition of Very late antigen 4/vascular cell adhesion molecule 1 interaction in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Cell Culture Conditions: CHO-K1 cells previously transfected with G-alpha 16 were subsequently transfected with the human CRTH2 receptor and the neom...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in RamosMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Cell Culture Conditions: CHO-K1 cells previously transfected with G-alpha 16 were subsequently transfected with the human CRTH2 receptor and the neom...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 0.420nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 0.420nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.480nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Cell Culture Conditions: CHO-K1 cells previously transfected with G-alpha 16 were subsequently transfected with the human CRTH2 receptor and the neom...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in RamosMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair