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Found 132 with Last Name = 'bailey' and Initial = 'k'
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461458(CHEMBL4229200)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461462(CHEMBL4225786)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461457(CHEMBL4225963)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461454(CHEMBL4224936)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461450(CHEMBL4226720)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461451(CHEMBL4226523)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461463(CHEMBL4225442)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461453(CHEMBL4226984)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461468(CHEMBL4227243)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50461456(CHEMBL4228095)
Affinity DataKi: <6.31E+3nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
The University of Edinburgh

LigandPNGBDBM85116(Cyclophilin Inhibitor, 15 | Cyclophilin Inhibitor,...)
Affinity DataKi:  6.80E+3nMAssay Description:The promising ligand from the results obtained from ESI-MS assay are subjected to PPIase in vitro assay. The PPIase assay assesses the abil9ity of l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
The University of Edinburgh

LigandPNGBDBM85118(Cyclophilin Inhibitor, 3d)
Affinity DataKi: >1.00E+5nMAssay Description:The promising ligand from the results obtained from ESI-MS assay are subjected to PPIase in vitro assay. The PPIase assay assesses the abil9ity of l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
The University of Edinburgh

LigandPNGBDBM85117(Cyclophilin Inhibitor, 3c)
Affinity DataKi: >1.00E+5nMAssay Description:The promising ligand from the results obtained from ESI-MS assay are subjected to PPIase in vitro assay. The PPIase assay assesses the abil9ity of l...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
The University of Edinburgh

LigandPNGBDBM85115(Cyclophilin Inhibitor, 3a)
Affinity DataKi: >1.00E+5nMAssay Description:The promising ligand from the results obtained from ESI-MS assay are subjected to PPIase in vitro assay. The PPIase assay assesses the abil9ity of l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
The University of Edinburgh

LigandPNGBDBM85116(Cyclophilin Inhibitor, 15 | Cyclophilin Inhibitor,...)
Affinity DataKi: >1.00E+5nMAssay Description:The promising ligand from the results obtained from ESI-MS assay are subjected to PPIase in vitro assay. The PPIase assay assesses the abil9ity of l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
The University of Edinburgh

LigandPNGBDBM85119(Cyclophilin Inhibitor, 3e)
Affinity DataKi:  2.07E+5nMAssay Description:The promising ligand from the results obtained from ESI-MS assay are subjected to PPIase in vitro assay. The PPIase assay assesses the abil9ity of l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282823(2-Butyl-6-(1-hydroxy-1-methyl-2-pyrrolidin-2-yl-et...)
Affinity DataIC50:  3.5nMAssay Description:Compound was tested for in vitro for AII receptor antagonistic activity in bovine adrenal cortex.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50212952(CHEMBL46150)
Affinity DataIC50:  5nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50049207(2-Butyl-6-(1-methoxy-1-methyl-ethyl)-3-[2'-(1H-tet...)
Affinity DataIC50:  6nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50212954(CHEMBL295114)
Affinity DataIC50:  11nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282897(2-Butyl-6-(5R,8S)-7-oxa-1-aza-bicyclo[3.2.1]oct-8-...)
Affinity DataIC50:  16nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282821(2-Butyl-6-((2S,3aR)-2-methyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  17nMAssay Description:Binding affinity of the compound expressed as inhibitory concentration towards bovine adrenal cortex angiotensin II receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282821(2-Butyl-6-((2S,3aR)-2-methyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  17nMAssay Description:Binding affinity expressed as inhibitory concentration against angiotensin II receptor of rat adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282805(2-Butyl-6-((2R,3aR)-2-methyl-hexahydro-isoxazolo[2...)
Affinity DataIC50:  22nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282821(2-Butyl-6-((2S,3aR)-2-methyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  26nMAssay Description:Binding affinity expressed as inhibitory concentration against angiotensin II receptor of rat adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282821(2-Butyl-6-((2S,3aR)-2-methyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  27nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50009718(2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetrazol-5-yl)-biph...)
Affinity DataIC50:  27nMAssay Description:Compound was tested for in vitro for AII receptor antagonistic activity in bovine adrenal cortex.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282792(2-Butyl-6-((2S,3aR)-2-methyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  27nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282794(5-{2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  30nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282881(2-Butyl-6-(1-methoxy-1-methyl-ethyl)-3-[2'-(1H-tet...)
Affinity DataIC50:  31nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50049207(2-Butyl-6-(1-methoxy-1-methyl-ethyl)-3-[2'-(1H-tet...)
Affinity DataIC50:  31nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282798(2-Butyl-6-(2S,3aR)-hexahydro-pyrrolo[1,2-b]isoxazo...)
Affinity DataIC50:  32nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282888(2-Butyl-6-((2S,3aS,8aR)-6,6-dimethyl-octahydro-fur...)
Affinity DataIC50:  32nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282806(2-Butyl-6-((2S,3aR)-2-hydroxymethyl-hexahydro-pyrr...)
Affinity DataIC50:  35nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282821(2-Butyl-6-((2S,3aR)-2-methyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  38nMAssay Description:Binding affinity of the compound expressed as inhibitory concentration towards bovine adrenal cortex angiotensin II receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282802(2-Butyl-6-(2S,3aR)-hexahydro-isoxazolo[2,3-a]pyrid...)
Affinity DataIC50:  38nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282898(2-Butyl-6-((1S,3aR,8aS,8bR)-6,6-dimethyl-octahydro...)
Affinity DataIC50:  38nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282821(2-Butyl-6-((2S,3aR)-2-methyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  38nMAssay Description:Binding affinity of the compound expressed as inhibitory concentration towards bovine adrenal cortex angiotensin II receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282818(2-Butyl-6-((2S,3aR)-6,6-dimethyl-hexahydro-pyrrolo...)
Affinity DataIC50:  39nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282893(2-Butyl-6-(6R,8S)-9-oxa-1-aza-bicyclo[4.2.1]non-8-...)
Affinity DataIC50:  42nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282886(2-Butyl-6-((3S,3aS,6aS)-2-methyl-4-oxo-hexahydro-c...)
Affinity DataIC50:  42nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282896(2-Butyl-6-((3R,5R)-5-hydroxymethyl-2-methyl-isoxaz...)
Affinity DataIC50:  43nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50212953(CHEMBL47914)
Affinity DataIC50:  44nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282807((2S,3aR)-2-{2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)...)
Affinity DataIC50:  46nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50212951(CHEMBL47449)
Affinity DataIC50:  47nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282808(2-Butyl-6-((2S,3aR)-2-methyl-hexahydro-isoxazolo[2...)
Affinity DataIC50:  47nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282901(2-Butyl-6-((3R,3aS,8aR,8bS)-6,6-dimethyl-octahydro...)
Affinity DataIC50:  53nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282791(2-Butyl-6-((2R,3aR)-2-methyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  55nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282892(2-Butyl-6-(3,3a,4,5,6,7-hexahydro-pyrazolo[1,5-a]p...)
Affinity DataIC50:  56nMAssay Description:In vitro binding affinity to angiotensin II receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282813(2-Butyl-6-((2R,3aR)-2-phenyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  56nMAssay Description:In vitro Angiotensin II receptor antagonism in bovine adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
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