BindingDB PrimarySearch_ki

Found 130 with Last Name = 'pickard' and Initial = 'l'

Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385915(CHEMBL2042135)

IC50: 22nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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3D Structure (crystal)

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526266(CHEMBL4565193)

IC50: 27nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526281(CHEMBL4576457)

IC50: 33nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385916(CHEMBL2042136)

IC50: 37nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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3D Structure (crystal)

Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385922(CHEMBL2042035)

IC50: 47nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385923(CHEMBL2042036)

IC50: 47nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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CHEMBL PC cid PC sid Similars

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Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385924(CHEMBL2042037)

IC50: 58nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385916(CHEMBL2042136)

IC50: 59nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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3D Structure (crystal)

Glycogen synthase kinase-3 beta(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385915(CHEMBL2042135)

IC50: 70nMAssay Description:Inhibition of GSK3beta incubated for 30 mins prior to substrate addition study done at apparent ATP Km for enzymeMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526267(CHEMBL4444939)

IC50: 72nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385914(CHEMBL2042042)

IC50: 73nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526277(CHEMBL4588737)

IC50: 80nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526266(CHEMBL4565193)

IC50: 87nMAssay Description:Displacement for LanthaScreen tracer from dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) ATP binding site KEN domain after 60 mi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526278(CHEMBL4453631)

IC50: 90nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385928(CHEMBL2042038)

IC50: 93nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526269(CHEMBL4516160)

IC50: 100nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Tyrosine-protein kinase Lck(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385915(CHEMBL2042135)

IC50: 110nMAssay Description:Inhibition of LCK incubated for 30 mins prior to substrate addition study done at apparent ATP Km for enzymeMore data for this Ligand-Target Pair

PDB Reactome pathway
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526267(CHEMBL4444939)

IC50: 110nMAssay Description:Displacement for LanthaScreen tracer from dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) ATP binding site KEN domain after 60 mi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526280(CHEMBL4534769)

IC50: 110nMAssay Description:Displacement for LanthaScreen tracer from dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) ATP binding site KEN domain after 60 mi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385919(CHEMBL2042031)

IC50: 120nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526280(CHEMBL4534769)

IC50: 122nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526279(CHEMBL4450996)

IC50: 130nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526282(CHEMBL4530582)

IC50: 130nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526278(CHEMBL4453631)

IC50: 130nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526281(CHEMBL4576457)

IC50: 140nMAssay Description:Displacement for LanthaScreen tracer from dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) ATP binding site KEN domain after 60 mi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526269(CHEMBL4516160)

IC50: 150nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526281(CHEMBL4576457)

IC50: 150nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526284(CHEMBL4568715)

IC50: 160nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526277(CHEMBL4588737)

IC50: 160nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526273(CHEMBL4538288)

IC50: 160nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526273(CHEMBL4538288)

IC50: 170nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526279(CHEMBL4450996)

IC50: 180nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526280(CHEMBL4534769)

IC50: 190nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526271(CHEMBL4468785)

IC50: 190nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526275(CHEMBL4515949)

IC50: 200nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385913(CHEMBL2042032)

IC50: 210nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526270(CHEMBL4554474)

IC50: 218nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
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3D Structure (crystal)

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526266(CHEMBL4565193)

IC50: 240nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526271(CHEMBL4468785)

IC50: 250nMAssay Description:Displacement for LanthaScreen tracer from dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) ATP binding site KEN domain after 60 mi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526277(CHEMBL4588737)

IC50: 270nMAssay Description:Displacement for LanthaScreen tracer from dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) ATP binding site KEN domain after 60 mi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM192719(KIRA analog, 1)

IC50: 290nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526287(CHEMBL4525939)

IC50: 303nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385929(CHEMBL2042039)

IC50: 318nMAssay Description:Inhibition of Nek2 using 5-FAM-KKLNRTLSVA-COOH as substrate after 1 hr by caliper methodMore data for this Ligand-Target Pair

PDB Reactome pathway
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526267(CHEMBL4444939)

IC50: 320nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526269(CHEMBL4516160)

IC50: 330nMAssay Description:Displacement for LanthaScreen tracer from dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) ATP binding site KEN domain after 60 mi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase D2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL

PNG

BDBM50385915(CHEMBL2042135)

IC50: 330nMAssay Description:Inhibition of PKD2 incubated for 30 mins prior to substrate addition study done at apparent ATP Km for enzymeMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526278(CHEMBL4453631)

IC50: 390nMAssay Description:Displacement for LanthaScreen tracer from dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) ATP binding site KEN domain after 60 mi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM192719(KIRA analog, 1)

IC50: 400nMAssay Description:Displacement for LanthaScreen tracer from dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) ATP binding site KEN domain after 60 mi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM192719(KIRA analog, 1)

IC50: 450nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) -dependent cleavage of FAM-labeled stem-loop RNA containing the XBP...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University of Leicester

Curated by ChEMBL

PNG

BDBM50526284(CHEMBL4568715)

IC50: 470nMAssay Description:Inhibition of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin) autophosphorylation at S724 after 25 mins in presence of ATP by dis...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
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Displayed 1 to 50 (of 130 total ) | Next | Last >>

Filter my 130 hits

Targets 15▿
- Serine/threonine-protein kinase/endoribonuclease IRE1 78
- Serine/threonine-protein kinase Nek2 21
- Serine/threonine-protein kinase PLK1 10
- Cyclin-dependent kinase 2 4
- Dual specificity protein kinase TTK 4
- Aurora kinase A 4
- Serine/threonine-protein kinase Chk2 1
- Tyrosine-protein kinase Lck 1
- Serine/threonine-protein kinase D2 1
- Tyrosine-protein kinase ABL1 1
- Hepatocyte growth factor receptor 1
- Proto-oncogene tyrosine-protein kinase Src 1
- Tyrosine-protein kinase Fyn 1
- Tyrosine-protein kinase Lyn 1
- Glycogen synthase kinase-3 beta 1
Publications 2▿
- J Med Chem 62: 2447-2465 (2019) 78
- J Med Chem 55: 3228-41 (2012) 52
Institutions 2▿
- University of Leicester 78
- The Institute Of Cancer Research 52
Affinity: 22 to 5.0E+4 nM▿
- IC50 129
- EC50 1
- Affinity ≤ nM
Xtal structures: 3
Docked structures: 0
Catalog Cmpds: 5