TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 0.220nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 0.360nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 0.590nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 0.940nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 0.980nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 0.990nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of MAO-A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 6.90nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 7.40nMAssay Description:Inhibition of GSK3alpha (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of DYRK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of electric eel AChE using acetylcholine chloride as substrate incubated measured after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of BuChE (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of DYRK3 (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 122nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human BACE1 in human SH-SY5Y cells using fluorogenic 7-methoxycoumarin-4-yl)acetyl-Ser-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-ArgL...More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human BACE1 in human SH-SY5Y cells using fluorogenic 7-methoxycoumarin-4-yl)acetyl-Ser-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-ArgL...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 142nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 142nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 208nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 216nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 221nMAssay Description:Inhibition of GSK3beta (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 225nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant human BACE1 using fluorogenic 7-methoxycoumarin-4-yl)acetyl-Ser-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-ArgLys(2, 4-dinitrophenyl)-...More data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of recombinant human BACE1 using fluorogenic 7-methoxycoumarin-4-yl)acetyl-Ser-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-ArgLys(2, 4-dinitrophenyl)-...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 535nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of electric eel AChE incubated measured after 25 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Louisiana At Lafayette
Curated by ChEMBL
University Of Louisiana At Lafayette
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of amyloid beta 1 to 42 aggregation in human SH-SY5Y cellsMore data for this Ligand-Target Pair
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