Affinity DataKi: 17nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Binding affinity to human 5HT4More data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
Affinity DataKi: 437nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
Affinity DataKi: 596nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University of Arizona
Curated by ChEMBL
University of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:The concentration that inhibits 50% specific binding was determined against the Melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University of Arizona
Curated by ChEMBL
University of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:The concentration that inhibits 50% specific binding was determined against the Melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.790nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University of Arizona
Curated by ChEMBL
University of Arizona
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:The concentration that inhibits 50% specific binding was determined against the Melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 169nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
Affinity DataIC50: 364nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 820nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.88E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.18E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.05E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 4.25E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 4.53E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University of Arizona
Curated by ChEMBL
University of Arizona
Curated by ChEMBL
Affinity DataEC50: 0.150nMAssay Description:Effective concentration against Melanocortin 1 receptor transfected into L-cells was determined by concentration of peptide for 50% maximal cAMP gene...More data for this Ligand-Target Pair