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Found 118 with Last Name = 'macdonald' and Initial = 'm'
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325659(8-fluoro-N-phenyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325661(8-fluoro-N-propyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi:  384nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325663(CHEMBL1224035 | N-butyl-8-fluoro-3,3a,4,9b-tetrahy...)
Affinity DataKi:  489nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325660(8-fluoro-N-isopropyl-3,3a,4,9b-tetrahydro-1H-thioc...)
Affinity DataKi:  569nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325664(CHEMBL1224036 | N-phenyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325667(CHEMBL1224103 | N-cyclohexyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi:  1.77E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325670(CHEMBL1224106 | N-o-tolyl-3,3a,4,9b-tetrahydro-1H-...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325659(8-fluoro-N-phenyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi:  5.17E+3nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325666(CHEMBL1224102 | N-propyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi:  6.60E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325664(CHEMBL1224036 | N-phenyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325665(CHEMBL1224101 | N-isopropyl-3,3a,4,9b-tetrahydro-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Citalopram from human SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325665(CHEMBL1224101 | N-isopropyl-3,3a,4,9b-tetrahydro-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325666(CHEMBL1224102 | N-propyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325666(CHEMBL1224102 | N-propyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325667(CHEMBL1224103 | N-cyclohexyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325667(CHEMBL1224103 | N-cyclohexyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325668(CHEMBL1224104 | N-tert-butyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325668(CHEMBL1224104 | N-tert-butyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325668(CHEMBL1224104 | N-tert-butyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325669(CHEMBL1224105 | N-butyl-3,3a,4,9b-tetrahydro-1H-ch...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325669(CHEMBL1224105 | N-butyl-3,3a,4,9b-tetrahydro-1H-ch...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325669(CHEMBL1224105 | N-butyl-3,3a,4,9b-tetrahydro-1H-ch...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325670(CHEMBL1224106 | N-o-tolyl-3,3a,4,9b-tetrahydro-1H-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325670(CHEMBL1224106 | N-o-tolyl-3,3a,4,9b-tetrahydro-1H-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]WIN-3542 from human DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Nisoxetine from human NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325664(CHEMBL1224036 | N-phenyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325663(CHEMBL1224035 | N-butyl-8-fluoro-3,3a,4,9b-tetrahy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325663(CHEMBL1224035 | N-butyl-8-fluoro-3,3a,4,9b-tetrahy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325661(8-fluoro-N-propyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325661(8-fluoro-N-propyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325660(8-fluoro-N-isopropyl-3,3a,4,9b-tetrahydro-1H-thioc...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325660(8-fluoro-N-isopropyl-3,3a,4,9b-tetrahydro-1H-thioc...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325659(8-fluoro-N-phenyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325665(CHEMBL1224101 | N-isopropyl-3,3a,4,9b-tetrahydro-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39156(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(2-hydroxy...)
Affinity DataIC50:  240nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313364((2S,3R,4R,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylphen...)
Affinity DataIC50:  250nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39146(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-[2-(2-hydr...)
Affinity DataIC50:  300nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39124(3-chloranyl-1-(3,4-dichlorophenyl)-4-(dimethylamin...)
Affinity DataIC50:  300nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39146(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-[2-(2-hydr...)
Affinity DataIC50:  400nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39124(3-chloranyl-1-(3,4-dichlorophenyl)-4-(dimethylamin...)
Affinity DataIC50:  400nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313335(6-(cyclohexylamino)-N-(4-sulfamoylphenyl)pyrimidin...)
Affinity DataIC50:  450nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM34194(3-chloranyl-1-(3,4-dichlorophenyl)-4-(4-methylpipe...)
Affinity DataIC50:  600nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39147(3-chloranyl-1-(3,4-dichlorophenyl)-4-[(3R)-3-methy...)
Affinity DataIC50:  600nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39156(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(2-hydroxy...)
Affinity DataIC50:  620nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-related protein A1(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39149(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-[(E)-3-phe...)
Affinity DataIC50:  690nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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