Affinity DataKi: 260nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+3nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.80E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.90E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.20E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.40E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.50E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.60E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.80E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.60E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 9.80E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.14E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore
Curated by ChEMBL
University Of Mysore
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore
Curated by ChEMBL
University Of Mysore
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore
Curated by ChEMBL
University Of Mysore
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore
Curated by ChEMBL
University Of Mysore
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 185nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 186nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 192nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 195nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore
Curated by ChEMBL
University Of Mysore
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore
Curated by ChEMBL
University Of Mysore
Curated by ChEMBL
Affinity DataIC50: 312nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 318nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 325nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 362nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 362nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore
Curated by ChEMBL
University Of Mysore
Curated by ChEMBL
Affinity DataIC50: 365nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 368nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore
Curated by ChEMBL
University Of Mysore
Curated by ChEMBL
Affinity DataIC50: 388nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 392nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair