Affinity DataKi: 0.790nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [125I]-NDP-R-MSH from melanocortin receptor 1 in mouse B16F10 cells after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Antagonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of MTII from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of Eu-NDP-MSH from human MC1R expressed in HEK293T cells after 2 hrs by DELFIA methodMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Antagonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Antagonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Antagonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Displacement of [125I]-NDP-R-MSH from mouse melanocortin receptor 4 expressed in HEK293 cells after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Antagonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Antagonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Antagonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of MTII from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of MTII from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Antagonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Antagonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation incubated ...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Displacement of MTII from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair