TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Cincinnati
Curated by ChEMBL
University Of Cincinnati
Curated by ChEMBL
Affinity DataKi: 0.00600nMAssay Description:Binding affinity towards human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Compound was evaluated to inhibit the thrombin enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Compound was evaluated to inhibit the thrombin enzymeMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Cincinnati
Curated by ChEMBL
University Of Cincinnati
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity towards human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Binding affinity towards human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.850nMAssay Description:Compound was evaluated to inhibit the thrombin enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Binding affinity towards human melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Compound was evaluated to inhibit the thrombin enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Cincinnati
Curated by ChEMBL
University Of Cincinnati
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:In vitro agonist potency was evaluated in HEK293 cells transfected with human melanocortin receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Compound was evaluated to inhibit the thrombin enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity to thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity towards human melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity to MC4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Cincinnati
Curated by ChEMBL
University Of Cincinnati
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Binding affinity towards human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Cincinnati
Curated by ChEMBL
University Of Cincinnati
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Binding affinity towards human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding affinity to thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:In vitro agonist potency was evaluated in HEK293 cells transfected with human melanocortin receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of europium-labeled NDP-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity to thrombinMore data for this Ligand-Target Pair