TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 460nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 860nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity towards human Corticotropin releasing factor receptor 1 by the displacement of [125I]-CRF from CHO cellsMore data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Nanjing University of Science and Technology
Curated by ChEMBL
Nanjing University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte BuChE using S-butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding affinity to biotinylated Keap1 DC domain (unknown origin) by biolayer interferometry assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of Nrf2-mediated ARE activity in human HepG2-ARE-C8 cells after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 3.60nMAssay Description:Binding affinity to biotinylated Keap1 DC domain (unknown origin) by biolayer interferometry assayMore data for this Ligand-Target Pair
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 26nMAssay Description:Binding affinity to recombinant human Keap1 Kelch domain (321 to 609) expressed in Escherichia coli BL21(DE3)pLysS cells after 30 mins by fluorescenc...More data for this Ligand-Target Pair
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