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Found 37 with Last Name = 'tomioka' and Initial = 'n'
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064089(4-hydroxymethyl-7,10-diisopropyl-8,10,13-trimethyl...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064090((S)-2-Decyl-5-hydroxymethyl-1-methyl-1,4,5,6-tetra...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073876((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-met...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064092(5'-hydroxymethyl-2'-isopropyl-1',4,4-trimethyl-(2'...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073875((1S,4S,5aS,9aS)-1,7,7-Tributyl-4-hydroxymethyl-5a-...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064094(5'-hydroxymethyl-2'-isopropyl-1'-methyl-(2'S,5'S)-...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073873((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-1,5a-d...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057510((2S,5S)-8-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064093((7S,10S)-10-Hydroxymethyl-7-isopropyl-4,4,6-trimet...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073878((4R,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073872((4S,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073870((4R,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073871((4R,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073877((4S,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057513((2S,5S)-5-Hydroxymethyl-2-isopropyl-1-methyl-1,4,5...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064088((7S,10S)-10-Hydroxymethyl-7-isopropyl-1,1,6-trimet...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064095((7S,10S)-10-Hydroxymethyl-7-isopropyl-1,1,4,4,6-pe...)
Affinity DataKi:  5.10E+3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099669(CHEMBL295139 | Succinic acid benzyl ester 3-carbox...)
Affinity DataIC50:  210nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099672(CHEMBL50599 | Succinic acid 3-carboxymethyl-1-(4-c...)
Affinity DataIC50:  310nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099675(CHEMBL416825 | Succinic acid 3-carboxymethyl-1-(4-...)
Affinity DataIC50:  540nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099667(5-Methyl-4-oxo-hexanoic acid 3-carboxymethyl-1-(4-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099673(5-Methyl-hexanoic acid 3-carboxymethyl-1-(4-chloro...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099671(CHEMBL48119 | Heptanoic acid 3-carboxymethyl-1-(4-...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50029074(2-{1-[(4-chlorophenyl)carbonyl]-5-hydroxy-2-methyl...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099674(CHEMBL47836 | [1-(4-Chloro-benzoyl)-5-(2-hydroxy-e...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099677(CHEMBL417723 | [1-(4-Chloro-benzoyl)-5-(3-hydroxy-...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099666(CHEMBL48025 | {4-[3-(4-Fluoro-3-nitro-phenyl)-urei...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099676(4-[(2-Amino-4-hydroxy-pteridin-6-ylmethyl)-(2,2,2-...)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099665(6-amino-2-[(hydrazinocarbonyl)amino]-1,3-dioxo-2,3...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099678(2-Bromo-5-methoxy-thiobenzoic acid S-[1-(3-chloro-...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099668(3-(4-Bromo-2-chloro-phenylcarbamoyl)-acrylic acid ...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50099670(2-(4-(4-aminophenylsulfonyl)phenylamino)acetic aci...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Aldose reductase (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed