Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 34nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 460nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 810nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 850nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 9.20E+3nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.05E+4nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Center For Bio-Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.50E+4nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]NECA in rat striatal membraneMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Rattus norvegicus)
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Affinity DataIC50: 6.72E+3nMAssay Description:Inhibition of Wistar rat heart SERCA2a after 1 hrMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(RAT)
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Affinity DataIC50: 8.23E+3nMAssay Description:Inhibition of Wistar rat kidney Na+,K+-ATPase alpha1 after 2 hrsMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rattus norvegicus)
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of Wistar rat EDL muscle SERCA1a after 1 hrMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 10nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 0.200nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 0.200nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 3.15E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 7.50E+3nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 9.65E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 1.03E+5nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 3.21E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair