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Found 152 with Last Name = 'andreasen' and Initial = 'pa'
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataKi:  6.80nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  8nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  9.90nMAssay Description:Inhibition of human wild-type plasma kallikrein catalytic domain after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  14nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataKi:  15nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataKi:  20nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataKi:  20nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  22nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Mus musculus)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  27nMAssay Description:Inhibition of mouse plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  32nMAssay Description:Inhibition of human plasma kallikrein catalytic domain E217A mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Mus musculus)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  43nMAssay Description:Inhibition of mouse plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  45nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Mus musculus)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  50nMAssay Description:Inhibition of mouse plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  54nMAssay Description:Inhibition of human plasma kallikrein catalytic domain G99Y mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499242(CHEMBL3736473)
Affinity DataKi:  64nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  136nMAssay Description:Inhibition of human plasma kallikrein catalytic domain G99Y mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  166nMAssay Description:Inhibition of human plasma kallikrein catalytic domain E217R mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  201nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataKi:  246nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataKi:  340nMAssay Description:Inhibition of human uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM23891(3-amidinophenylalanine deriv., 35 | CHEMBL107955 |...)
Affinity DataKi:  370nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  384nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM23891(3-amidinophenylalanine deriv., 35 | CHEMBL107955 |...)
Affinity DataKi:  500nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499239(CHEMBL3734777)
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM23891(3-amidinophenylalanine deriv., 35 | CHEMBL107955 |...)
Affinity DataKi:  650nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  833nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataKi:  903nMAssay Description:Inhibition of human uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  907nMAssay Description:Inhibition of human wild-type plasma kallikrein catalytic domain after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  938nMAssay Description:Inhibition of human plasma kallikrein catalytic domain E217A mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM23891(3-amidinophenylalanine deriv., 35 | CHEMBL107955 |...)
Affinity DataKi:  980nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM23891(3-amidinophenylalanine deriv., 35 | CHEMBL107955 |...)
Affinity DataKi:  1.46E+3nMAssay Description:Inhibition of plasmin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  1.58E+3nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  1.69E+3nMAssay Description:Inhibition of human plasma kallikrein catalytic domain E217R mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataKi:  1.77E+3nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM23891(3-amidinophenylalanine deriv., 35 | CHEMBL107955 |...)
Affinity DataKi:  2.51E+3nMAssay Description:Inhibition of tPA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  2.56E+3nMAssay Description:Inhibition of human coagulation factor 11a after 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Mus musculus)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  2.97E+3nMAssay Description:Inhibition of mouse plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Mus musculus)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  3.42E+3nMAssay Description:Inhibition of mouse plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Mus musculus)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  3.67E+3nMAssay Description:Inhibition of mouse plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  3.97E+3nMAssay Description:Inhibition of human coagulation factor 11a after 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Mus musculus)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  4.61E+3nMAssay Description:Inhibition of mouse plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  6.63E+3nMAssay Description:Inhibition of human coagulation factor 11a after 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  9.80E+3nMAssay Description:Inhibition of human plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  1.06E+4nMAssay Description:Inhibition of human plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  1.21E+4nMAssay Description:Inhibition of human coagulation factor 11a after 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  1.25E+4nMAssay Description:Inhibition of human plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  1.41E+4nMAssay Description:Inhibition of bovine beta-trypsin after 15 mins using Bz-Ile-Glu(g-OR)-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  1.45E+4nMAssay Description:Inhibition of bovine beta-trypsin after 15 mins using Bz-Ile-Glu(g-OR)-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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