Affinity DataKi: 36nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 730nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 830nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: >2.10E+3nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Antagonist activity at human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+3nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.60E+3nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 12nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 16nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 16nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 17nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 17nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 18nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 21nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 24nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 24nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 26nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 29nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 33nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 39nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 39nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 42nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 48nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 51nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
Institute of Cancer Research
US Patent
Institute of Cancer Research
US Patent
Affinity DataIC50: 76nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair