Affinity DataKi: 0.330nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 2(Homo sapiens (Human))
University of Virginia
Curated by PDSP Ki Database
University of Virginia
Curated by PDSP Ki Database
TargetLeukotriene B4 receptor 2(Homo sapiens (Human))
University of Virginia
Curated by PDSP Ki Database
University of Virginia
Curated by PDSP Ki Database
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Addiction Research Foundation
Curated by PDSP Ki Database
Addiction Research Foundation
Curated by PDSP Ki Database
Affinity DataKi: 7.40nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [3H]-ZM241385 from wild type human adenosine receptor A2a expressed in HEK293 cell membranes after 240 mins by scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
Affinity DataKi: 40nMAssay Description:Displacement of [3H]PSB-603 from human A2B receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]PSB-11 from human A3 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
Affinity DataKi: 68nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Addiction Research Foundation
Curated by PDSP Ki Database
Addiction Research Foundation
Curated by PDSP Ki Database
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
Affinity DataKi: 112nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Addiction Research Foundation
Curated by PDSP Ki Database
Addiction Research Foundation
Curated by PDSP Ki Database
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataKi: 146nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
Affinity DataKi: 288nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 347nMAssay Description:Displacement of [3H]PSB-11 from human A3 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 372nMAssay Description:Displacement of [3H]PSB-603 from human A2B receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
Affinity DataKi: 417nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 562nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Addiction Research Foundation
Curated by PDSP Ki Database
Addiction Research Foundation
Curated by PDSP Ki Database
TargetLeukotriene B4 receptor 2(Homo sapiens (Human))
University of Virginia
Curated by PDSP Ki Database
University of Virginia
Curated by PDSP Ki Database
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
Affinity DataKi: 1.02E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+3nMAssay Description:Displacement of [3H]PSB-11 from human A3 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Addiction Research Foundation
Curated by PDSP Ki Database
Addiction Research Foundation
Curated by PDSP Ki Database
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Addiction Research Foundation
Curated by PDSP Ki Database
Addiction Research Foundation
Curated by PDSP Ki Database
Affinity DataKi: 1.35E+3nMAssay Description:Displacement of [3H]PSB-11 from human A3 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Addiction Research Foundation
Curated by PDSP Ki Database
Addiction Research Foundation
Curated by PDSP Ki Database
Affinity DataKi: 2.69E+3nMAssay Description:Displacement of [3H]PSB-11 from human A3 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database
The Centre For Addiction and Mental Health
Curated by PDSP Ki Database