Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0620nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.254nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Negative logarithm causing 50% receptor occupancy against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Inhibition constant against serotonin transporterMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Negative logarithm causing 50% receptor occupancy against beta-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Negative logarithm causing 50% receptor occupancy against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibitory concentration against angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibitory concentration against angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
Affinity DataKi: 0.960nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition constant against alpha adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition constant against angiotensin I converting enzymeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Msd
Curated by ChEMBL
Msd
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Inhibition of human ERG by dofetilide binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Inhibition constant against serotonin transporterMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Negative logarithm causing 50% receptor occupancy against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibitory concentration against endothelin receptor type AMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition constant against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of the Collagenase enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair