TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.0170nMAssay Description:Displacement of [3H]paroxetine from serotonin transporter of rat cerebral cortexMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 0.0340nMAssay Description:Compound was evaluated for its ability to inhibit Striatal Dopamine Receptor in rat brain through radioreceptor assay carried out with agonist ligand...More data for this Ligand-Target Pair
Affinity DataKi: 0.0530nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0530nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:Ability to displace [3H]- paroxetine from Serotonin transporter in rat cerebral cortical homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Research Biochemicals International
Curated by ChEMBL
Research Biochemicals International
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:In vitro binding affinity towards dopamine transporter in rat striatal membranes by [3H]GBR-12395 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.0620nMAssay Description:Binding affinity to serotonin transporter (SERT) in rat forebrain tissueMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:In vitro binding affinity towards serotonin transporter in rat cerebral cortical homogenates by [3H]paroxetine displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [3H]paroxetine from serotonin transporter of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Compound was evaluated for affinity towards dopamine D1-like receptor in homogenate of caudateputamen tissue from rat brainMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:In vitro binding affinity towards serotonin transporter in rat cerebral cortical homogenates by [3H]paroxetine displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]paroxetine from serotonin transporter of rat cerebral cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Research Biochemicals International
Curated by ChEMBL
Research Biochemicals International
Curated by ChEMBL
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]paroxetine from SERT in rat frontoparietal cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]-cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity of compound for Serotonin transporter with [3H]- paroxetine as radioligand in corpus striatum tissue from rat forebrainMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:In vitro binding affinity of compound for Serotonin transporter with [3H]- paroxetine as radioligand in corpus striatum tissue from rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Dopamine receptor D2 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Displacement of [3H]paroxetine from serotonin transporter of rat cerebral cortexMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Agonist activity was tested in vitro against Dopamine receptor from rat brain membranes with [3H]ADT-6,7-dihydroxy-2-aminotetralin]More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]-cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Compound was evaluated for its ability to inhibit Dopamine receptor D2 in rat striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Dopamine receptor D2 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Compound was evaluated for affinity towards dopamine D1-like receptor in homogenate of caudateputamen tissue from rat brainMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Research Biochemicals International
Curated by ChEMBL
Research Biochemicals International
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:In vitro binding affinity towards serotonin transporter in rat cerebral cortical homogenates by [3H]paroxetine displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:In vitro binding affinity of compound for Serotonin transporter with [3H]- paroxetine as radioligand in corpus striatum tissue from rat forebrainMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:In vitro binding affinity towards serotonin transporter in rat cerebral cortical homogenates by [3H]paroxetine displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]paroxetine from SERT in rat frontoparietal cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.380nMAssay Description:Displacement of [3H]paroxetine from serotonin transporter of rat cerebral cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Binding affinity to serotonin transporter (SERT) in rat forebrain tissueMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H]paroxetine from SERT in rat frontoparietal cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Dopamine receptor D2 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.440nMAssay Description:In vitro binding affinity of compound for Serotonin transporter with [3H]- paroxetine as radioligand in corpus striatum tissue from rat forebrainMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]8-OH-DPAT from rat 5HT1A receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:In vitro binding affinity towards serotonin transporter in rat cerebral cortical homogenates by [3H]paroxetine displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Affinity for Serotonin transporter by displacing [3H]-Paroxetine from rat forebrainMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Displacement of [3H]cyanoimipramine from SERT in rat cerebral cortex homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Ability to displace [3H]- paroxetine from Serotonin transporter in rat cerebral cortical homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Displacement of [3H]paroxetine from serotonin transporter of rat cerebral cortexMore data for this Ligand-Target Pair