Affinity DataKi: 610nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIAMore data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIAMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 2.23E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.99E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 3.82E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.82E+3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIAMore data for this Ligand-Target Pair
Affinity DataKi: 4.54E+3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIAMore data for this Ligand-Target Pair
Affinity DataKi: 4.54E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.40E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.40E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 1.12E+4nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+4nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 1.75E+4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+4nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.50E+4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 5.55E+4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 5.71E+4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 1.89E+5nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Agonistic activity against adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+5nMAssay Description:Displacement of [3H]DPCPX from rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Agonistic activity against adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+5nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+5nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataEC50: >100nMAssay Description:[S]GTP gamma-S binding against adenosine A1 receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataEC50: 6.44E+3nMAssay Description:Binding against human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Binding against human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 869nMAssay Description:Binding against human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.23E+3nMAssay Description:[S]GTP gamma-S binding against adenosine A1 receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataEC50: 59nMAssay Description:Binding against human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Kd value for adenosine A1 receptor binding at 14.5 uMMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Kd value for adenosine A1 receptor binding at 145 uMMore data for this Ligand-Target Pair
Affinity DataEC50: 87nMAssay Description:[S]GTP gamma-S binding against adenosine A1 receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Binding against Human Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:[S]GTP gamma-S binding against adenosine A1 receptor in rat brainMore data for this Ligand-Target Pair