Affinity DataKi: 0.0500nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute Of Organic Synthesis
Curated by ChEMBL
Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]DTG from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 760nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 860nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 3.20E+3nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.90E+3nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.40E+3nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.40E+3nMAssay Description:Binding affinity towards Melanocortin 3 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 4.50E+3nMAssay Description:Binding affinity towards Melanocortin 3 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Binding affinity towards Melanocortin 5 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Binding affinity towards Melanocortin 3 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 5.60E+3nMAssay Description:Binding affinity towards Melanocortin 3 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 6.50E+3nMAssay Description:Binding affinity towards Melanocortin 3 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Binding affinity towards Melanocortin 3 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 8.20E+3nMAssay Description:Binding affinity towards Melanocortin 5 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 8.80E+3nMAssay Description:Binding affinity towards Melanocortin 3 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 9.80E+3nMAssay Description:Binding affinity towards Melanocortin 5 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Binding affinity towards Melanocortin 5 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of factor 12a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Binding affinity towards Melanocortin 3 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of factor 12a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of factor 12a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of factor 12a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of factor 12a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of factor 12a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of factor 12a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+4nMAssay Description:Binding affinity towards Melanocortin 5 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+4nMAssay Description:Binding affinity towards Melanocortin 5 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+4nMAssay Description:Binding affinity towards Melanocortin 5 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Binding affinity towards Melanocortin 5 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+4nMAssay Description:Binding affinity towards Melanocortin 3 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair