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Found 285 with Last Name = 'madapa' and Initial = 's'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]Way100635 from human recombinant 5-HT1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210757(CHEMBL3921278)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210764(CHEMBL3976659)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210759(CHEMBL3905947)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50599264(CHEMBL5204813)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210767(CHEMBL3945691)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210761(CHEMBL3961827)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152837(CHEMBL595489)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50378584(STEPHOLIDINE)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152842(CHEMBL3780268)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210754(CHEMBL3982215)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152846(CHEMBL3780506)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210763(CHEMBL3894329)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50089979(CHEMBL3581250)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152845(CHEMBL3781840)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210756(CHEMBL3975220)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152847(CHEMBL3779928)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210762(CHEMBL3954556)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152841(CHEMBL3780184)
Affinity DataKi:  12nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152841(CHEMBL3780184)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152845(CHEMBL3781840)
Affinity DataKi:  13nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152836(CHEMBL3780481)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50090078(CHEMBL3581245)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in HEK cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50599254(CHEMBL5174366)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50599252(CHEMBL5180016)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5-HT2A receptor expressed in HEKT cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210754(CHEMBL3982215)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]N-methylspiperone from human D2 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50152844(CHEMBL3780140)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50250422((+)-N-methyl-laurotetanine | CHEMBL464099 | N-meth...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in HEK cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50060417(5-Methyl-3,5-dihydro-2H-pyrrolo[2,3-f]indole-1-car...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50089974(CHEMBL3581254)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in HEK cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50599263(CHEMBL5195241)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50599264(CHEMBL5204813)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50089976(CHEMBL3581252)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in HEK cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50089980(CHEMBL3581249)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50210758(CHEMBL3945856)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]N-methylspiperone from human D2 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50089973(CHEMBL3581255)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in HEK cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50599263(CHEMBL5195241)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation...More data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50089979(CHEMBL3581250)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in HEK cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50090077(CHEMBL3580670)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in HEK cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50599259(CHEMBL5203303)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50090001(CHEMBL3581248)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in HEK cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50089976(CHEMBL3581252)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
City University Of New York

Curated by ChEMBL
LigandPNGBDBM50378584(STEPHOLIDINE)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]N-methylspiperone from human D3 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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