Affinity DataIC50: 1nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Petersburg State University
Curated by ChEMBL
Saint Petersburg State University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human ERG expressed in cell membranes after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate by fluorescent inhibitor screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albuminMore data for this Ligand-Target Pair