TargetDisintegrin and metalloproteinase domain-containing protein 17 [215-477,S266A,N452Q](Homo sapiens (Human))
Schering-Plough Research Institute
Schering-Plough Research Institute
Affinity DataKi: 0.0600nM ΔG°: -57.8kJ/molepH: 7.3 T: 2°CAssay Description:Enzyme activity was determined by a kinetic assay measuring the rate of increase in fluorescent intensity generated by the cleavage of an internally ...More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17 [215-477,S266A,N452Q](Homo sapiens (Human))
Schering-Plough Research Institute
Schering-Plough Research Institute
Affinity DataKi: 0.140nM ΔG°: -55.7kJ/molepH: 7.3 T: 2°CAssay Description:Enzyme activity was determined by a kinetic assay measuring the rate of increase in fluorescent intensity generated by the cleavage of an internally ...More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17 [215-477,S266A,N452Q](Homo sapiens (Human))
Schering-Plough Research Institute
Schering-Plough Research Institute
Affinity DataKi: 0.180nM ΔG°: -55.1kJ/molepH: 7.3 T: 2°CAssay Description:Enzyme activity was determined by a kinetic assay measuring the rate of increase in fluorescent intensity generated by the cleavage of an internally ...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17 [215-477,S266A,N452Q](Homo sapiens (Human))
Schering-Plough Research Institute
Schering-Plough Research Institute
Affinity DataKi: 3nM ΔG°: -48.2kJ/molepH: 7.3 T: 2°CAssay Description:Enzyme activity was determined by a kinetic assay measuring the rate of increase in fluorescent intensity generated by the cleavage of an internally ...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair