Affinity DataKi: 1.40E+3nMAssay Description:Competitive inhibition of recombinant Trypanosoma cruzi cruzain by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Competitive inhibition of recombinant Trypanosoma cruzi cruzain by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Mixed inhibition of recombinant Trypanosoma brucei rhodesain expressed in Pichia pastoris by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+4nMAssay Description:Competitive inhibition of recombinant Trypanosoma cruzi cruzain in presence of varying levels of Z-phe-Arg-amidomethylcoumarin substrate by Lineweave...More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins without preincubation by f...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of human recombinant glutathione reductase using glutathione as substrate preincubated for 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain expressed in Pichia pastoris using Z-FR-AMC as substrate preincubated for 10 mins followed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins without preincubation by f...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-phe-Arg-amidomethylcoumarin as substrate by fluorometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-phe-Arg-amidomethylcoumarin as substrate by fluorometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins without preincubation by f...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-phe-Arg-amidomethylcoumarin as substrate by fluorometric methodMore data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain expressed in Pichia pastoris using Z-FR-AMC as substrate and measured at 12 sec interval for 5...More data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain expressed in Pichia pastoris using Z-FR-AMC as substrate preincubated for 10 mins followed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-phe-Arg-amidomethylcoumarin as substrate by fluorometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-phe-Arg-amidomethylcoumarin as substrate by fluorometric methodMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: 4.58E+4nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain expressed in Pichia pastoris using Z-FR-AMC as substrate and measured at 12 sec interval for 5...More data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-phe-Arg-amidomethylcoumarin as substrate by fluorometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant glutathione reductase using glutathione as substrate preincubated for 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase expressed in Escherichia coli BL21(DE3) assessed as reduction of oxidized trypanothione prein...More data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant glutathione reductase using glutathione as substrate preincubated for 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant glutathione reductase using glutathione as substrate preincubated for 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant glutathione reductase using glutathione as substrate preincubated for 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant glutathione reductase using glutathione as substrate preincubated for 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant glutathione reductase using glutathione as substrate preincubated for 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant glutathione reductase using glutathione as substrate preincubated for 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Universidade Federal De Minas Gerais
Curated by ChEMBL
Universidade Federal De Minas Gerais
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant glutathione reductase using glutathione as substrate preincubated for 30 mins by colorimetric assayMore data for this Ligand-Target Pair