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Found 196 with Last Name = 'bonn' and Initial = 't'
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81961(CAS_124393-85-7 | SHX | silahexocyclium)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81959(CAS_115-63-9 | Hexocyclium)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81961(CAS_124393-85-7 | SHX | silahexocyclium)
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81961(CAS_124393-85-7 | SHX | silahexocyclium)
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81959(CAS_115-63-9 | Hexocyclium)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81959(CAS_115-63-9 | Hexocyclium)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81961(CAS_124393-85-7 | SHX | silahexocyclium)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81959(CAS_115-63-9 | Hexocyclium)
Affinity DataKi:  3.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50010101(2-(diethylamino)ethyl 1-cyclohexylcyclohexanecarbo...)
Affinity DataKi:  5.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81959(CAS_115-63-9 | Hexocyclium)
Affinity DataKi:  5.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81960(CAS_113010-69-8 | HHD | hexahydrodifenidol)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)
Affinity DataKi:  12.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81960(CAS_113010-69-8 | HHD | hexahydrodifenidol)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Karo Pharma

Curated by ChEMBL
LigandPNGBDBM50466897(CHEMBL4287715)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from human N-terminal 6His-tagged-RORC2 LBD (259 to 483 residues) expressed in Escherichia coli (DE3) cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Karo Pharma

Curated by ChEMBL
LigandPNGBDBM50466891(CHEMBL4281109)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from human N-terminal 6His-tagged-RORC2 LBD (259 to 483 residues) expressed in Escherichia coli (DE3) cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81959(CAS_115-63-9 | Hexocyclium)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81961(CAS_124393-85-7 | SHX | silahexocyclium)
Affinity DataKi:  35nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)
Affinity DataKi:  44nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Karo Pharma

Curated by ChEMBL
LigandPNGBDBM50466893(CHEMBL4291727)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from human N-terminal 6His-tagged-RORC2 LBD (259 to 483 residues) expressed in Escherichia coli (DE3) cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  57nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81960(CAS_113010-69-8 | HHD | hexahydrodifenidol)
Affinity DataKi:  83nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  88nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  107nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  118nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  186nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81960(CAS_113010-69-8 | HHD | hexahydrodifenidol)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50010101(2-(diethylamino)ethyl 1-cyclohexylcyclohexanecarbo...)
Affinity DataKi:  244nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)
Affinity DataKi:  249nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of The West Indies

Curated by ChEMBL
LigandPNGBDBM50423775(CHEMBL602321)
Affinity DataKi:  747nMAssay Description:Displacement of [3H]flunitrezepam from GABA-A alpha-1-beta-2-gamma-2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  820nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  838nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  906nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Karo Pharma

Curated by ChEMBL
LigandPNGBDBM50466892(CHEMBL4283871)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from human N-terminal 6His-tagged-RORC2 LBD (259 to 483 residues) expressed in Escherichia coli (DE3) cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  1.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  2.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  2.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Homo sapiens (Human))
University Of The West Indies

Curated by ChEMBL
LigandPNGBDBM50423775(CHEMBL602321)
Affinity DataKi:  8.08E+3nMAssay Description:Displacement of [3H]flunitrezepam from GABA-A alpha-2-beta-2-gamma-2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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