TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
City University Of New York
Curated by ChEMBL
City University Of New York
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
City University Of New York
Curated by ChEMBL
City University Of New York
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
City University Of New York
Curated by ChEMBL
City University Of New York
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]N-methylspiperone from human D2 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting metho...More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]N-methylspiperone from human D2 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting metho...More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to dopamine D3 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]N-methylspiperone from human D3 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting metho...More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [3H]N-methylspiperone from human D3 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting metho...More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by PDSP assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
City University Of New York
Curated by ChEMBL
City University Of New York
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]SCH2390 from human dopamine D1 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [3H]N-methylspiperone from human D2 receptor expressed in HEKT cell membranes after 90 mins by microbeta scintillation counting metho...More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by PDSP assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
City University Of New York
Curated by ChEMBL
City University Of New York
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair