Compile Data Set for Download or QSAR
maximum 50k data
Found 173 with Last Name = 'yue' and Initial = 'x'
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108979(CHEMBL3597316)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108980(CHEMBL3597317)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108983(CHEMBL3597320)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108978(CHEMBL3597315)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108986(CHEMBL3597324)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108981(CHEMBL3597318)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108984(CHEMBL3597321)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108984(CHEMBL3597321)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108978(CHEMBL3597315)
Affinity DataKi:  13nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108982(CHEMBL3597319)
Affinity DataKi:  29nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108982(CHEMBL3597319)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataKi:  74nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108985(CHEMBL3597322)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108986(CHEMBL3597324)
Affinity DataKi:  191nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108983(CHEMBL3597320)
Affinity DataKi:  821nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108979(CHEMBL3597316)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108981(CHEMBL3597318)
Affinity DataKi:  8.64E+3nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108980(CHEMBL3597317)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108984(CHEMBL3597321)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108984(CHEMBL3597321)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University

Curated by ChEMBL
LigandPNGBDBM50108985(CHEMBL3597322)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of KDR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50210697(CHEMBL3962233)
Affinity DataIC50:  1nMAssay Description:Inhibition of N-terminal GST-tagged human EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus expression system preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50210747(CHEMBL3968039)
Affinity DataIC50:  1nMAssay Description:Inhibition of N-terminal GST-tagged human EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus expression system preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50507551(CHEMBL4587222)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of Ron (unknown origin) using FAM-labelled peptide and ATP incubated for 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of Ron (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Shanghai Institute Of Materia Medica (Simm)

Curated by ChEMBL
LigandPNGBDBM50436850(CERITINIB | CHEMBL2403108 | LDK378 | US10053458, C...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523921(CHEMBL4446992)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  11nMAssay Description:Inhibition of N-terminal GST-tagged human EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus expression system preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Shanghai Institute Of Materia Medica (Simm)

Curated by ChEMBL
LigandPNGBDBM50025759(CHEMBL3330859)
Affinity DataIC50:  12nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50210748(CHEMBL3920551)
Affinity DataIC50:  14nMAssay Description:Inhibition of N-terminal GST-tagged human VEGFR-2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50210705(CHEMBL3979264)
Affinity DataIC50:  14nMAssay Description:Inhibition of N-terminal GST-tagged human EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus expression system preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50210695(CHEMBL3929448)
Affinity DataIC50:  14nMAssay Description:Inhibition of N-terminal GST-tagged human VEGFR-2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  15nMAssay Description:Inhibition of N-terminal GST-tagged human VEGFR-2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50210752(CHEMBL3938494)
Affinity DataIC50:  15nMAssay Description:Inhibition of N-terminal GST-tagged human EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus expression system preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50507551(CHEMBL4587222)
Affinity DataIC50:  15nMAssay Description:Inhibition of c-Met (unknown origin) using FAM-labelled peptide and ATP incubated for 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50210701(CHEMBL3957025)
Affinity DataIC50:  17nMAssay Description:Inhibition of N-terminal GST-tagged human EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus expression system preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Shanghai Institute Of Materia Medica (Simm)

Curated by ChEMBL
LigandPNGBDBM50025760(CHEMBL3330858)
Affinity DataIC50:  18nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50210698(CHEMBL3939588)
Affinity DataIC50:  18nMAssay Description:Inhibition of N-terminal GST-tagged human VEGFR-2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  19nMAssay Description:Inhibition of c-MET (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523921(CHEMBL4446992)
Affinity DataIC50:  19nMAssay Description:Inhibition of VEGFR2 (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  19nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50025779(CHEMBL3330850)
Affinity DataIC50:  20nMAssay Description:Inhibition of purified c-MET (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  21nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  21nMAssay Description:Inhibition of KDR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  29nMAssay Description:Inhibition of [125I]VCAM-Ig binding to VLA-4 of Jurkat cells in the presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297565(CHEMBL4160512)
Affinity DataIC50:  30nMAssay Description:In vitro antiviral activity against HIV-1 Reverse transcriptase M184V mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297346(CHEMBL4167741)
Affinity DataIC50:  37nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 173 total ) | Next | Last >>
Jump to: