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Found 54 with Last Name = 'hirasawa' and Initial = 'y'
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50199522((+)-huperzine A | (+-)-HA | (-)-1-Amino-13-ethylid...)
Affinity DataIC50:  53nMAssay Description:Inhibition of bovine acetylcholinesteraseMore data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308527(10-methoxy-N(1)-methylburnamine-17-O-veratrate | C...)
Affinity DataIC50:  500nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308533(CHEMBL589254 | Methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308529(CHEMBL589220 | Methyl (14E)-19-[(benzoyloxy)methyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50483304(11-Epi-Tubulysin D)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50483306(CHEBI:80036 | Tubulysin D)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50483305(13-Epi-Tubulysin D)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308528(Alstiphyllanine D | CHEMBL540945)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308527(10-methoxy-N(1)-methylburnamine-17-O-veratrate | C...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308532((14E)-14-ethylidene-6-methoxy-19-(methoxycarbonyl)...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50201171((1S,9R)-1-amino-13-[2-hydroxy-eth-(E)-ylidene]-11-...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of bovine erythrocyte acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308528(Alstiphyllanine D | CHEMBL540945)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308531((14E)-19-{[(3,4-dimethoxyphenyl)carbonyloxy]methyl...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308533(CHEMBL589254 | Methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50483307(CHEMBL1643767)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308530(CHEMBL602442 | Methyl (14E)-14-ethylidene-6-hydrox...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50201170(CHEMBL241838 | carinatumins B (2))
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of bovine erythrocyte acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308532((14E)-14-ethylidene-6-methoxy-19-(methoxycarbonyl)...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308535(CHEMBL601712 | methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308529(CHEMBL589220 | Methyl (14E)-19-[(benzoyloxy)methyl...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50316419(CHEMBL1097908 | Gneyulin B)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of SGLT2 transfected in african green monkey COS1 cells assessed as alpha-D-[U-14C]glucopyranoside uptake after 30 mins by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50223709(CHEMBL240094 | cryptadine B)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of bovine acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50271482(CHEMBL455781 | lycoparin C)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of acetylcholinesterase from bovine erythrocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50316418(CHEMBL1097907 | Gneyulin A)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of SGLT2 transfected in african green monkey COS1 cells assessed as alpha-D-[U-14C]glucopyranoside uptake after 30 mins by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50316418(CHEMBL1097907 | Gneyulin A)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of SGLT1 transfected in african green monkey COS1 cells assessed as alpha-D-[U-14C]glucopyranoside uptake after 30 mins by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308526(Burnamine-17-O-3',4',5'-trimethoxybenzoate | CHEMB...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308531((14E)-19-{[(3,4-dimethoxyphenyl)carbonyloxy]methyl...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50316419(CHEMBL1097908 | Gneyulin B)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of SGLT1 transfected in african green monkey COS1 cells assessed as alpha-D-[U-14C]glucopyranoside uptake after 30 mins by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308525(Alstiphyllanine F | CHEMBL592521)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308524(Alstiphyllanine E | CHEMBL592477)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308525(Alstiphyllanine F | CHEMBL592521)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308524(Alstiphyllanine E | CHEMBL592477)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308526(Burnamine-17-O-3',4',5'-trimethoxybenzoate | CHEMB...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308530(CHEMBL602442 | Methyl (14E)-14-ethylidene-6-hydrox...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308534(CHEMBL590530 | methyl (14E)-19-[(acetyloxy)methyl]...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308535(CHEMBL601712 | methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  9.70E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50321281(Alpneumine C | CHEMBL1163798)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50321282(Alpneumine D | CHEMBL1163799)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50321283(Alpneumine E | CHEMBL1163800)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50321284(Alpneumine F | CHEMBL1165402)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50321285(Alpneumine G | CHEMBL1164480)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50321280(Alpneumine B | CHEMBL1164346)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308536(CHEMBL590772 | methyl (14E)-19-[(benzyloxy)methyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50321286(Alpneumine H | CHEMBL1165844)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308534(CHEMBL590530 | methyl (14E)-19-[(acetyloxy)methyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50201172((4aS,5S,7S,8aS)-7-methyl-5-(1-oxy-3,4,5,6-tetrahyd...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of bovine erythrocyte acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308536(CHEMBL590772 | methyl (14E)-19-[(benzyloxy)methyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50321287(Alpneumine A | CHEMBL1164076)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mushroom tyrosinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM20875(1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihyd...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
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