Affinity DataKi: 0.380nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 231nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 247nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 367nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:The compound was tested for inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.47E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:The inhibitory constant(Ki) for MTA phosphorylase activity was determined by using a mouse liver enzyme preparationMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:The inhibitory constant(Ki) for MTA phosphorylase activity was determined by using a mouse liver enzyme preparationMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:The inhibitory constant(Ki) for MTA phosphorylase activity was determined by using a mouse liver enzyme preparationMore data for this Ligand-Target Pair
Affinity DataKi: 3.29E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:The inhibitory constant(Ki) for MTA phosphorylase activity was determined by using a mouse liver enzyme preparationMore data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 6.50E+3nMAssay Description:The inhibitory constant(Ki) for MTA phosphorylase activity was determined by using a mouse liver enzyme preparationMore data for this Ligand-Target Pair
Affinity DataKi: 7.04E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 9.04E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 9.80E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:The inhibitory constant(Ki) for MTA phosphorylase activity was determined by using a mouse liver enzyme preparationMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+4nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 1.42E+4nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 1.71E+4nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:The inhibitory constant(Ki) for MTA phosphorylase activity was determined by using a mouse liver enzyme preparationMore data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Biotech Research Institute
Curated by ChEMBL
Biotech Research Institute
Curated by ChEMBL
Affinity DataKi: 2.72E+4nMAssay Description:The compound was tested for inhibitory activity against tissue plasminogen activatorMore data for this Ligand-Target Pair
Affinity DataKi: 4.79E+4nMAssay Description:The compound was tested for inhibitory activity against human plasminMore data for this Ligand-Target Pair
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institute Of Science & Technology
Curated by ChEMBL
Institute Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against human plasma mu-calpainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institute Of Science & Technology
Curated by ChEMBL
Institute Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibitory concentration against human plasma mu-calpainMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institute Of Science & Technology
Curated by ChEMBL
Institute Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibitory concentration against human plasma mu-calpainMore data for this Ligand-Target Pair
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institute Of Science & Technology
Curated by ChEMBL
Institute Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibitory concentration against human plasma mu-calpainMore data for this Ligand-Target Pair
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institute Of Science & Technology
Curated by ChEMBL
Institute Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibitory concentration against human plasma mu-calpainMore data for this Ligand-Target Pair