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Found 53 with Last Name = 'akue-gedu' and Initial = 'r'
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  10nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299245(7-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  40nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  120nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299247(1-(1,10-Dihydropyrrolo[2,3-a]carbazol-3-yl)-2,2,2-...)
Affinity DataIC50:  170nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299250(7-(2,4-Difluorophenyl)-1,10-dihydropyrrolo[2,3-a]c...)
Affinity DataIC50:  200nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299248(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carboxamide ...)
Affinity DataIC50:  210nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM50295872(5-Iodo-4-(1-Methyl-1H-indol-3-yl)pyrimidin-2-amine...)
Affinity DataIC50:  400nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299246(7-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole | CHEM...)
Affinity DataIC50:  440nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  510nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299245(7-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  570nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295874(4-(1H-indol-3-yl)-5-(4-(trifluoromethyl)phenyl)pyr...)
Affinity DataIC50:  580nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295873(4-[2-Amino-4-(1H-indol-3-yl)pyrimidin-5-yl]benzami...)
Affinity DataIC50:  580nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295875(4-(1H-Indol-3-yl)-5-(3-methoxyphenyl)pyrimidin-2-a...)
Affinity DataIC50:  600nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295876(4-(1H-Indol-3-yl)-5-(3-aminophenyl)pyrimidin-2-ami...)
Affinity DataIC50:  640nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299250(7-(2,4-Difluorophenyl)-1,10-dihydropyrrolo[2,3-a]c...)
Affinity DataIC50:  660nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Centre National De La Recherche Scientifique

US Patent
LigandPNGBDBM50299248(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carboxamide ...)
Affinity DataIC50:  780nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM50295877(4-[2-Amino-4-(1-methyl-1H-indol-3-yl)pyrimidin-5-y...)
Affinity DataIC50:  900nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295878(4-(1-Methyl-1H-indol-3-yl)-5-(pyridin-4-yl)pyrimid...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295879(4-(1-Methyl-1H-indol-3-yl)-5-(3-aminophenyl)pyrimi...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295873(4-[2-Amino-4-(1H-indol-3-yl)pyrimidin-5-yl]benzami...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295880(4-[2-Amino-4-(1-methyl-1H-indol-3-yl)pyrimidin-5-y...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295874(4-(1H-indol-3-yl)-5-(4-(trifluoromethyl)phenyl)pyr...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295878(4-(1-Methyl-1H-indol-3-yl)-5-(pyridin-4-yl)pyrimid...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295872(5-Iodo-4-(1-Methyl-1H-indol-3-yl)pyrimidin-2-amine...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295881(4-(1H-indol-3-yl)-5-(4-(trifluoromethoxy)phenyl)py...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295882(4-(1-Methyl-1H-indol-3-yl)-5-(3-methoxyphenyl)pyri...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295875(4-(1H-Indol-3-yl)-5-(3-methoxyphenyl)pyrimidin-2-a...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295883(4-(1-Methyl-1H-indol-3-yl)-5,50-bipyrimidin-2-amin...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295881(4-(1H-indol-3-yl)-5-(4-(trifluoromethoxy)phenyl)py...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295872(5-Iodo-4-(1-Methyl-1H-indol-3-yl)pyrimidin-2-amine...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295884(1-(4-(2-amino-4-(1-methyl-1H-indol-3-yl)pyrimidin-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295878(4-(1-Methyl-1H-indol-3-yl)-5-(pyridin-4-yl)pyrimid...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295876(4-(1H-Indol-3-yl)-5-(3-aminophenyl)pyrimidin-2-ami...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295880(4-[2-Amino-4-(1-methyl-1H-indol-3-yl)pyrimidin-5-y...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295882(4-(1-Methyl-1H-indol-3-yl)-5-(3-methoxyphenyl)pyri...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295881(4-(1H-indol-3-yl)-5-(4-(trifluoromethoxy)phenyl)py...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295884(1-(4-(2-amino-4-(1-methyl-1H-indol-3-yl)pyrimidin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295885(5-(biphenyl-4-yl)-4-(1-methyl-1H-indol-3-yl)pyrimi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295875(4-(1H-Indol-3-yl)-5-(3-methoxyphenyl)pyrimidin-2-a...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295883(4-(1-Methyl-1H-indol-3-yl)-5,50-bipyrimidin-2-amin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295876(4-(1H-Indol-3-yl)-5-(3-aminophenyl)pyrimidin-2-ami...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295879(4-(1-Methyl-1H-indol-3-yl)-5-(3-aminophenyl)pyrimi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295873(4-[2-Amino-4-(1H-indol-3-yl)pyrimidin-5-yl]benzami...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295880(4-[2-Amino-4-(1-methyl-1H-indol-3-yl)pyrimidin-5-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295877(4-[2-Amino-4-(1-methyl-1H-indol-3-yl)pyrimidin-5-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295883(4-(1-Methyl-1H-indol-3-yl)-5,50-bipyrimidin-2-amin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295885(5-(biphenyl-4-yl)-4-(1-methyl-1H-indol-3-yl)pyrimi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295884(1-(4-(2-amino-4-(1-methyl-1H-indol-3-yl)pyrimidin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295885(5-(biphenyl-4-yl)-4-(1-methyl-1H-indol-3-yl)pyrimi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295882(4-(1-Methyl-1H-indol-3-yl)-5-(3-methoxyphenyl)pyri...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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