TargetTissue alpha-L-fucosidase(Bos taurus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Ki value against bovine alpha-L-fucosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of human recombinant beta-glucocerebrosidase assessed as p-nitrophenolate accumulation preincubated for 10 mins before p-nitrophenyl-beta-...More data for this Ligand-Target Pair
TargetTissue alpha-L-fucosidase(Bos taurus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Inhibition of bovine epididymis alpha-L-fucosidase assessed as p-nitrophenol release by spectrophotometricallyMore data for this Ligand-Target Pair
TargetTissue alpha-L-fucosidase(Bos taurus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Ki value against bovine alpha-L-fucosidaseMore data for this Ligand-Target Pair
TargetTissue alpha-L-fucosidase(Bos taurus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of bovine epididymis alpha-L-fucosidase assessed as p-nitrophenol release by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibitory activity measured against alpha-L-fucosidase of bovine epididymis by colorimetric assay using the D-glucose oxidase-peroxidase methodMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibitory activity measured against alpha-L-fucosidase of bovine epididymis by colorimetric assay using the D-glucose oxidase-peroxidase methodMore data for this Ligand-Target Pair
TargetTissue alpha-L-fucosidase(Bos taurus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Ki value against bovine alpha-L-fucosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 200nM ΔG°: -39.8kJ/mole IC50: 270nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
Affinity DataKi: 280nM ΔG°: -38.9kJ/mole IC50: 500nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
Affinity DataKi: 300nM ΔG°: -38.7kJ/mole IC50: 660nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
Affinity DataKi: 420nM ΔG°: -37.9kJ/mole IC50: 820nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
TargetTissue alpha-L-fucosidase(Bos taurus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Ki value against bovine alpha-L-fucosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Compound was tested for binding affinity against alpha-glucosidaseMore data for this Ligand-Target Pair
TargetTissue alpha-L-fucosidase(Bos taurus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Inhibition of bovine epididymis alpha-L-fucosidase assessed as p-nitrophenol release by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Competitive inhibition of human lysosome alpha-galactosidase by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
Tohoku University School Of Medicine
Curated by ChEMBL
Tohoku University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nM ΔG°: -33.5kJ/mole IC50: 4.20E+3nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Inhibitory activity measured against alpha-L-fucosidase of bovine epididymis by colorimetric assay using the D-glucose oxidase-peroxidase methodMore data for this Ligand-Target Pair
TargetTissue alpha-L-fucosidase(Bos taurus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Ki value against bovine alpha-L-fucosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nM ΔG°: -31.2kJ/mole IC50: 1.30E+4nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
Affinity DataKi: 6.20E+3nMAssay Description:Compound was tested for binding affinity against alpha-glucosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.90E+3nMAssay Description:Compound was tested for binding affinity against alpha-glucosidaseMore data for this Ligand-Target Pair
TargetTissue alpha-L-fucosidase(Bos taurus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.40E+4nMAssay Description:Ki value against bovine alpha-L-fucosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+4nMAssay Description:Competitive Inhibitory activity against Golgi Alpha-mannosidase IIMore data for this Ligand-Target Pair
Affinity DataKi: <5.00E+4nMAssay Description:Competitive Inhibitory activity against Golgi Alpha-mannosidase IIMore data for this Ligand-Target Pair
Affinity DataKi: <5.00E+4nMAssay Description:Competitive Inhibitory activity against Golgi Alpha-mannosidase IIMore data for this Ligand-Target Pair
Affinity DataKi: <5.00E+4nMAssay Description:Competitive Inhibitory activity against Golgi Alpha-mannosidase IIMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+4nMAssay Description:Competitive Inhibitory activity against Golgi Alpha-mannosidase IIMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+4nM ΔG°: -24.4kJ/mole IC50: 2.40E+5nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+5nM ΔG°: -23.5kJ/mole IC50: 1.00E+5nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
Affinity DataKi: 1.16E+5nM ΔG°: -23.4kJ/mole IC50: 2.70E+5nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+5nMAssay Description:Competitive Inhibitory activity against Golgi Alpha-mannosidase IIMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+5nMAssay Description:Tested for competitive inhibition of golgi alpha mannosidase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMpH: 6.5Assay Description:Inhibition of coffee bean alpha-galactosidase assessed as p-nitrophenol release at pH 6.5 by spectrometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair