Affinity DataKi: 0.102nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.108nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Inhibition of human liver cathepsin B using Z-Phe-Arg-AMC as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.870nMAssay Description:Inhibition of rat ecto-5'-nucleotidase expressed in Sf9 cells by capillary electrophoresis methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Inhibition of rat ecto-5'-nucleotidase expressed in Sf9 cells by capillary electrophoresis methodMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: <1nMAssay Description:Inhibition of FITC-Bim binding to human His6-MPB tagged MCL1 expressed in Escherichia coli K-12 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.94nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human liver cathepsin B using Z-Phe-Arg-AMC as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 3.16nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of recombinant human cathepsin S expressed in insect cells using Z-Phe-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of human liver cathepsin B using Z-Phe-Arg-AMC as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 6.31nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 6.31nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 7.94nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 12.6nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibition of recombinant human cathepsin S expressed in insect cells using Z-Phe-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 14.1nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 19.9nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of recombinant human cathepsin K expressed in insect cells using Z-Leu-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of recombinant human cathepsin K expressed in insect cells using Z-Leu-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of recombinant human cathepsin S expressed in insect cells using Z-Phe-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of recombinant human cathepsin S expressed in insect cells using Z-Phe-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of recombinant human cathepsin S expressed in insect cells using Z-Phe-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of recombinant human cathepsin S expressed in insect cells using Z-Phe-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of recombinant human cathepsin K expressed in insect cells using Z-Leu-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of recombinant human cathepsin S expressed in insect cells using Z-Phe-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 39.8nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 39.8nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 39.8nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 39.8nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Inhibition of recombinant human cathepsin K expressed in insect cells using Z-Leu-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of recombinant human cathepsin S expressed in insect cells using Z-Phe-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of recombinant human cathepsin K expressed in insect cells using Z-Leu-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Inhibition of recombinant human cathepsin K expressed in insect cells using Z-Leu-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 45.3nMAssay Description:Inhibition of rat ecto-5'-nucleotidase expressed in Sf9 cells by capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 50.1nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universita£T
Curated by ChEMBL
Affinity DataKi: 50.1nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibition of recombinant human cathepsin K expressed in insect cells using Z-Leu-Arg-AMC as substrate measured after 60 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Inhibition of human recombinant matriptase catalytic domain expressed in HEK293 cells after 20 minsMore data for this Ligand-Target Pair