Affinity DataKi: 740nMAssay Description:Competitive inhibition of human MDH1 expressed in Escherichia coli using oxaloacetic acid as substrate in presence of NADH after 30 mins by double re...More data for this Ligand-Target Pair
Affinity DataKi: 950nMAssay Description:Inhibition of human MDH1 expressed in Escherichia coli after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Competitive inhibition of MDH2 (unknown origin) using varying NADH level by oxaloacetate-dependent NADH oxidation based Lineweaver-Burk plotMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Competitive inhibition of MDH2 (unknown origin) using varying NADH level by oxaloacetate-dependent NADH oxidation based Lineweaver-Burk plotMore data for this Ligand-Target Pair
Affinity DataIC50: 2.53nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.62nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 4.45nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of hypoxia-induced HIF1alpha transcriptional activity in human HeLa cells expressing HRE-Luc after 12 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
Affinity DataIC50: 14.8nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 16.9nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 17.7nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 20.3nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 23.8nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 25.9nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 28.5nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Gakushuin University
Curated by ChEMBL
Gakushuin University
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant KDR at 1 uM by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 32.6nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 32.7nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of hypoxia-induced HIF1alpha transcriptional activity in human HeLa cells expressing HRE-Luc after 12 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Gakushuin University
Curated by ChEMBL
Gakushuin University
Curated by ChEMBL
Affinity DataIC50: 65.5nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 87.1nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 106nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 214nMAssay Description:Inhibition of hypoxia-induced HIF1alpha transcriptional activity in human HeLa cells expressing HRE-Luc after 12 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of hypoxia-induced HIF1alpha transcriptional activity in human HeLa cells expressing HRE-Luc after 12 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Gakushuin University
Curated by ChEMBL
Gakushuin University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Gakushuin University
Curated by ChEMBL
Gakushuin University
Curated by ChEMBL
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Gakushuin University
Curated by ChEMBL
Gakushuin University
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of HIF-1alpha in human HCT116 cells incubated for 12 hrs under hypoxic conditions by HRE dual-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
Affinity DataIC50: 920nMAssay Description:Inhibition of human MDH1 expressed in Escherichia coli after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 940nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of human MDH2 after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human MDH1 expressed in Escherichia coli after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of HIF-1alpha in human HCT116 cells incubated for 12 hrs under hypoxic conditions by HRE dual-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of MDH1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of human MDH2 after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of human MDH2 after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of human MDH1 expressed in Escherichia coli after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human MDH1 expressed in Escherichia coli after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of human MDH1 expressed in Escherichia coli after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of human MDH2 after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of human MDH2 after 30 mins by oxaloacetate-dependent NADH oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of hypoxia-induced HIF1alpha transcriptional activity in human HeLa cells expressing HRE-Luc after 12 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of HIF-1alpha in human HCT116 cells incubated for 12 hrs under hypoxic conditions by HRE dual-luciferase reporter gene assayMore data for this Ligand-Target Pair