Affinity DataKi: 970nMAssay Description:Binding affinity to rat 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human muscarinic M1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human alpha2A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to rat alpha1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Binding affinity to human histamine H1 receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of dofetilide from hERGMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Compound was tested for its inhibitory activity against Matrix metalloproteinase-8 (MMP-8) in adjuvant arthritic rat model of rheumatoid arthritisMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Compound was tested for its inhibitory activity against Matrix metalloproteinase-9(MMP-9) in adjuvant arthritic rat model of rheumatoid arthritisMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Compound was tested for its inhibitory activity against Matrix metalloproteinase-8(MMP-8) in adjuvant arthritic rat model of rheumatoid arthritisMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Compound was tested for its inhibitory activity against Matrix Matrix metalloproteinase-9 in adjuvant arthritic rat model of rheumatoid arthritisMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Compound was tested for its inhibitory activity against Matrix metalloproteinase-8(MMP-8) in adjuvant arthritic rat model of rheumatoid arthritisMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Compound was tested for its inhibitory activity against Matrix metalloproteinase-9(MMP-9) in adjuvant arthritic rat model of rheumatoid arthritisMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of matrix metalloproteinase-3, MMP-3More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Compound was tested for its inhibitory activity against Matrix metalloproteinase-8 (MMP-8) in adjuvant arthritic rat model of rheumatoid arthritisMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Compound was tested for its inhibitory activity against Matrix metalloproteinase-8(MMP-8) in adjuvant arthritic rat model of rheumatoid arthritisMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of matrix metalloproteinase-8, MMP-8More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of matrix metalloproteinase-3, MMP-3More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Compound was tested for its inhibitory activity against Matrix metalloproteinase-9 in adjuvant arthritic rat model of rheumatoid arthritisMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of matrix metalloproteinase-9, MMP-9More data for this Ligand-Target Pair