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Found 294 with Last Name = 'bekhit' and Initial = 'aa'
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Alexandria

Curated by ChEMBL
LigandPNGBDBM50179019(3-benzyl-N-(2-morpholinoethyl)quinoxalin-2-amine |...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073539(CHEMBL3408926)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073512(CHEMBL3408911)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Alexandria

Curated by ChEMBL
LigandPNGBDBM50179021(3-(4-chlorobenzyl)-N-(2-morpholinoethyl)quinoxalin...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Alexandria

Curated by ChEMBL
LigandPNGBDBM50179017(1-(3-(4-chlorobenzyl)quinoxalin-2-yl)hydrazine | C...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50097456(CHEMBL3585822)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50378844(CHEMBL1258839)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50378846(CHEMBL1258610)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50378833(CHEMBL1257814)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Alexandria

Curated by ChEMBL
LigandPNGBDBM50088564(CHEMBL3577041)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50097459(CHEMBL3585817)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Alexandria

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073531(CHEMBL3408918)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of bovine brain mitochondria MAO-A by spectrofluorimetryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073533(CHEMBL3408920)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073532(CHEMBL3408919)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50378834(CHEMBL1257932)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073534(CHEMBL3408921)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50097463(CHEMBL3585814)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of bovine brain mitochondria MAO-B using benzylamine substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Alexandria

Curated by ChEMBL
LigandPNGBDBM50179020(2-(3-benzylquinoxalin-2-ylamino)ethanol | CHEMBL20...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50078676(CHEMBL3415443)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of bovine brain mitochondria MAO-A by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50078677(CHEMBL3415442)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of bovine brain mitochondria MAO-A by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50327216(3-Benzyl-2-(2-(2-chlorobenzylidene)hydrazinyl)quin...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50327220(4-Benzyl-1-(2-chlorophenyl)-[1,2,4]triazolo[4,3-a]...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50078679(CHEMBL3415439)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of bovine brain mitochondria MAO-A by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50327222(4-Benzoyl-1-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50327214(2-(2-(Benzo[d][1,3]dioxol-5-ylmethylene)hydrazinyl...)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073535(CHEMBL3408922)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50327221(4-Benzoyl-1-(3,4-dimethoxyphenyl)-[1,2,4]triazolo[...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073540(CHEMBL3408927)
Affinity DataIC50:  7.30nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Alexandria

Curated by ChEMBL
LigandPNGBDBM50179018(1-(3-benzyl-6,7-dichloroquinoxalin-2-yl)hydrazine ...)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50097460(CHEMBL3585818)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073536(CHEMBL3408923)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50378840(CHEMBL1258274)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Alexandria

Curated by ChEMBL
LigandPNGBDBM50179015(1-(3-benzylquinoxalin-2-yl)hydrazine | CHEMBL37967...)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50327223(4-Benzoyl-1-(3-bromo-4-(N,N-dimethylaminophenyl))-...)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50378839(CHEMBL1258160)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50327219(3-Benzyl-2-(2-(3-bromobenzylidene)hydrazinyl)quino...)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50093711(CHEMBL3585838)
Affinity DataIC50:  16nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Alexandria

Curated by ChEMBL
LigandPNGBDBM50088560(CHEMBL3577045)
Affinity DataIC50:  18nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50093778(CHEMBL3585828)
Affinity DataIC50:  18nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073537(CHEMBL3408924)
Affinity DataIC50:  22nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50378847(CHEMBL1258718)
Affinity DataIC50:  22nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50093779(CHEMBL3585827)
Affinity DataIC50:  28nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50378851(CHEMBL1257341)
Affinity DataIC50:  29nMAssay Description:Inhibition of MAOA by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50093710(CHEMBL3585839)
Affinity DataIC50:  32nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50097420(CHEMBL3585826)
Affinity DataIC50:  32nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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