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Found 61 with Last Name = 'bendale' and Initial = 'p'
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13321(1-Methyl-1H-imidazole-4-sulfonic Acid (2-Bromoally...)
Affinity DataIC50:  0.400nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13323(1-Methyl-1H-imidazole-4-sulfonic Acid Benzyl-[6-cy...)
Affinity DataIC50:  0.600nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13320(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  0.600nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13320(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  0.700nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13328(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  0.800nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13321(1-Methyl-1H-imidazole-4-sulfonic Acid (2-Bromoally...)
Affinity DataIC50:  0.800nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13319(BMS-386914 | CHEMBL183536 | [[6-Cyano-1-(3-methyl-...)
Affinity DataIC50:  0.900nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13325(4-{[[6-Cyano-1-(3-methyl-3H-imidazol-4-ylmethyl)-1...)
Affinity DataIC50:  1.10nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13319(BMS-386914 | CHEMBL183536 | [[6-Cyano-1-(3-methyl-...)
Affinity DataIC50:  1.20nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13322(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  1.20nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13323(1-Methyl-1H-imidazole-4-sulfonic Acid Benzyl-[6-cy...)
Affinity DataIC50:  1.20nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13331(N-tert-butyl-2-({6-isocyano-1-[(1-methyl-1H-imidaz...)
Affinity DataIC50:  1.40nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13324(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  1.5nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13322(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  1.5nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476682(CHEMBL428712 | PB-43)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13331(N-tert-butyl-2-({6-isocyano-1-[(1-methyl-1H-imidaz...)
Affinity DataIC50:  1.80nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476678(CHEMBL395222)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13327(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  2.80nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13328(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  3nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM13328(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  3nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13325(4-{[[6-Cyano-1-(3-methyl-3H-imidazol-4-ylmethyl)-1...)
Affinity DataIC50:  3.20nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476685(CHEMBL232104)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13324(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  3.40nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM13324(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM13327(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13327(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  3.80nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476680(CHEMBL234757)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM16180((2S)-2-{[4-({[(2S)-1-cyclohexyl-3-(ethylsulfanyl)p...)
Affinity DataIC50:  5nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13335(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  5nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM13335(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476679(CHEMBL232523)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13332(N-tert-Butyl-2-[[6-isocyano-1-(3-methyl-3H-imidazo...)
Affinity DataIC50:  6nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476681(CHEMBL234151 | PB-91)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476676(CHEMBL231662)
Affinity DataIC50:  7nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476675(CHEMBL233742)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13334(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  7.60nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476677(CHEMBL394086 | PB-90)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13335(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  8nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM16178(3-benzyl-1-(1H-imidazol-5-ylmethyl)-4-(thiophen-2-...)
Affinity DataIC50:  8nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM16181(1-[2-(4-cyanophenyl)-2-hydroxy-2-(1-methyl-1H-imid...)
Affinity DataIC50:  9nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13330(N-[(6-chloro-2,1,3-benzothiadiazol-5-yl)methyl]-N-...)
Affinity DataIC50:  10nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM13330(N-[(6-chloro-2,1,3-benzothiadiazol-5-yl)methyl]-N-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50:  15nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476674(CHEMBL394407 | PB-95)
Affinity DataIC50:  16nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM14434(6-[amino(4-chlorophenyl)(1-methyl-1H-imidazol-5-yl...)
Affinity DataIC50:  17nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13332(N-tert-Butyl-2-[[6-isocyano-1-(3-methyl-3H-imidazo...)
Affinity DataIC50:  25nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50476684(CHEMBL392237)
Affinity DataIC50:  25nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13326(1-Methyl-1H-imidazole-4-sulfonic Acid (1-Bromonaph...)
Affinity DataIC50:  28nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13334(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  42nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13330(N-[(6-chloro-2,1,3-benzothiadiazol-5-yl)methyl]-N-...)
Affinity DataIC50:  55nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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