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Found 105 with Last Name = 'benoist' and Initial = 'a'
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051495((S)-2-[(S)-2-(2-Hydroxy-acetyl)-pyrrolidine-1-carb...)
Affinity DataIC50:  0.100nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051520(CHEMBL305681 | [(2S,3aS,7aS)-2-(Pyrrolidine-1-carb...)
Affinity DataIC50:  0.900nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051511(CHEMBL80684 | [(1R,2S)-2-(4-Fluoro-phenyl)-cyclopr...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051523(((1R,2S)-2-Phenyl-cyclopropyl)-[(2S,3aS,7aS)-2-(py...)
Affinity DataIC50:  1.20nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051504(((1R,2S)-2-Phenyl-cyclopropyl)-[(2S,3aS,7aS)-2-(th...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051515(CHEMBL80698 | [(2S,3aS,7aS)-2-(Pyrrolidine-1-carbo...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051506(((1R,2S)-2-Phenyl-cyclopropyl)-[(S)-3-(pyrrolidine...)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051516(CHEMBL79213 | [(2S,3aS,7aS)-2-(Pyrrolidine-1-carbo...)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051508(CHEMBL75968 | [(2S,3aS,7aS)-2-(Isoxazolidine-2-car...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373665(CHEMBL442455)
Affinity DataIC50:  2nMAssay Description:Inhibition of NEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051489(((1R,2S)-2-Phenyl-cyclopropyl)-[(2S,3aS,7aS)-2-(py...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051483(CHEMBL80865 | [(2S,3aS,7aS)-2-(2,5-Dihydro-pyrrole...)
Affinity DataIC50:  2.40nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051544(CHEMBL311848 | [(2S,3aS,7aS)-2-(2,3-Dihydro-pyrrol...)
Affinity DataIC50:  2.70nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051513(((1R,2S)-2-Phenyl-cyclopropyl)-[(S)-3-(thiazolidin...)
Affinity DataIC50:  3.10nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051496(CHEMBL310228 | [(S)-3-(Pyrrolidine-1-carbonyl)-2-a...)
Affinity DataIC50:  3.20nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051537(CHEMBL80136 | [(1R,2S)-2-(4-Fluoro-phenyl)-cyclopr...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373657(CHEMBL450935)
Affinity DataIC50:  4nMAssay Description:Inhibition of NEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051543((2-Benzyl-cyclopropyl)-[(S)-3-(pyrrolidine-1-carbo...)
Affinity DataIC50:  4.20nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051484(CHEMBL307938 | [(S)-3-(Pyrrolidine-1-carbonyl)-2-a...)
Affinity DataIC50:  4.80nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051484(CHEMBL307938 | [(S)-3-(Pyrrolidine-1-carbonyl)-2-a...)
Affinity DataIC50:  4.80nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticamMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051488(((1R,2S)-2-Phenyl-cyclopropyl)-[(S)-3-(pyrrolidine...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051486(((1R,2S)-2-Naphthalen-2-yl-cyclopropyl)-[(S)-3-(py...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373663(CHEMBL273142)
Affinity DataIC50:  5nMAssay Description:Inhibition of NEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051518(6,6,6-Trifluoro-5-phenyl-1-[(2S,3aS,7aS)-2-(pyrrol...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051540((R)-3-(Pyrrolidine-1-carbonyl)-2-aza-bicyclo[2.2.1...)
Affinity DataIC50:  5.5nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50454200(CHEMBL2369824)
Affinity DataIC50:  5.5nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373668(CHEMBL270576)
Affinity DataIC50:  6nMAssay Description:Inhibition of NEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373661(CHEMBL257251)
Affinity DataIC50:  6nMAssay Description:Inhibition of NEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373660(CHEMBL255568)
Affinity DataIC50:  8nMAssay Description:Inhibition of NEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373664(CHEMBL409920)
Affinity DataIC50:  9nMAssay Description:Inhibition of NEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051487(5,5-Dicyclopropyl-1-[(S)-3-(pyrrolidine-1-carbonyl...)
Affinity DataIC50:  9nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373669(CHEMBL409720)
Affinity DataIC50:  10nMAssay Description:Inhibition of NEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051491(CHEMBL77149 | [(2S,3aS,7aS)-2-(3-Hydroxy-pyrrolidi...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051506(((1R,2S)-2-Phenyl-cyclopropyl)-[(S)-3-(pyrrolidine...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051481(CHEMBL306957 | [(1R,2S)-2-(4-Methoxy-phenyl)-cyclo...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051542(5,5-Dicyclopropyl-1-[(2S,3aS,7aS)-2-(pyrrolidine-1...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373659(CHEMBL258278)
Affinity DataIC50:  19nMAssay Description:Inhibition of NEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051536(6,6-Dicyclopropyl-1-[(S)-3-(pyrrolidine-1-carbonyl...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051512((R)-3-(2,5-Dihydro-pyrrole-1-carbonyl)-2-aza-bicyc...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051510((R)-3-(Pyrrolidine-1-carbonyl)-2-aza-bicyclo[2.2.2...)
Affinity DataIC50:  23nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373659(CHEMBL258278)
Affinity DataIC50:  23nMAssay Description:Inhibition of ACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051517((R)-3-(Thiazolidine-3-carbonyl)-2-aza-bicyclo[2.2....)
Affinity DataIC50:  24nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051546((E)-6,6-Dicyclopropyl-1-[(S)-3-(pyrrolidine-1-carb...)
Affinity DataIC50:  24nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051509(5,5-Dicyclopropyl-1-[(S)-3-(pyrrolidine-1-carbonyl...)
Affinity DataIC50:  26nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051505(4-Phenyl-1-[(R)-3-(pyrrolidine-1-carbonyl)-2-aza-b...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051479((3-Phenyl-cyclobutyl)-[(S)-3-(pyrrolidine-1-carbon...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Rattus norvegicus)
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051479((3-Phenyl-cyclobutyl)-[(S)-3-(pyrrolidine-1-carbon...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373665(CHEMBL442455)
Affinity DataIC50:  29nMAssay Description:Inhibition of ACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051550((3aS,7aS)-2-(Azetidine-1-carbonyl)-octahydro-indol...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Institut De Recherche Servier

Curated by ChEMBL
LigandPNGBDBM50051547((S)-2-(Pyrrolidine-1-carbonyl)-pyrrolidine-1-carbo...)
Affinity DataIC50:  32nMAssay Description:Inhibitory activity evaluated against Post-proline cleaving enzyme from Flavobacterium meningosepticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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