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Found 138 with Last Name = 'bera' and Initial = 'h'
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004462(CHEMBL3233329)
Affinity DataKi:  1.65E+3nMAssay Description:Mixed-type inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidide to thymine by Li...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004460(CHEMBL3233327)
Affinity DataKi:  1.77E+3nMAssay Description:Mixed-type inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidide to thymine by Li...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439105(CHEMBL2418061)
Affinity DataKi:  1.96E+4nMAssay Description:Mixed inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate by Lineweaver-Burk plot anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439106(CHEMBL2418074)
Affinity DataKi:  2.01E+4nMAssay Description:Mixed inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate by Lineweaver-Burk plot anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  10nMpH: 8.0 T: 2°CAssay Description:The in vitro AChE inhibitory activity was measured using the methods described earlier [Biochem. Pharmacol. 7:88-95]. Briefly, stock solutions (1mg/m...More data for this Ligand-Target Pair
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM20079(5-chloro-6-[(2-iminopyrrolidin-1-yl)methyl]-1,2,3,...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human placenta thymidine phosphorylase using [6-3H]dThd as substrate after 5 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM20079(5-chloro-6-[(2-iminopyrrolidin-1-yl)methyl]-1,2,3,...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human thymidine phosphorylaseMore data for this Ligand-Target Pair
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM20079(5-chloro-6-[(2-iminopyrrolidin-1-yl)methyl]-1,2,3,...)
Affinity DataIC50:  35nMAssay Description:Competitive inhibition of human thymidine phosphorylase in presence of thymidineMore data for this Ligand-Target Pair
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50443422(CHEMBL3087264)
Affinity DataIC50:  350nMAssay Description:Inhibition of human thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192120(2-(4-(1-benzoyl-3-(1H-indol-3-yl)-4,5-dihydro-1H-p...)
Affinity DataIC50:  680nMpH: 8.0 T: 2°CAssay Description:The in vitro AChE inhibitory activity was measured using the methods described earlier [Biochem. Pharmacol. 7:88-95]. Briefly, stock solutions (1mg/m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192116((3-(1H-indol-3-yl)-5-phenyl-4,5-dihydropyrazol-1-y...)
Affinity DataIC50:  740nMpH: 8.0 T: 2°CAssay Description:The in vitro AChE inhibitory activity was measured using the methods described earlier [Biochem. Pharmacol. 7:88-95]. Briefly, stock solutions (1mg/m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439105(CHEMBL2418061)
Affinity DataIC50:  2.95E+3nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Aimst University

Curated by ChEMBL
LigandPNGBDBM193765((E)-5-((2-(quinoxalin-2-yl)hydrazono)methyl)benzen...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of Escherichia coli K12 thymidine phosphorylase expressed in Escherichia coli preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004462(CHEMBL3233329)
Affinity DataIC50:  3.82E+3nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidine to thymine after 4 to 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004457(CHEMBL3233340)
Affinity DataIC50:  4.29E+3nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidine to thymine after 4 to 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004456(CHEMBL3233339)
Affinity DataIC50:  4.46E+3nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidine to thymine after 4 to 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004455(CHEMBL3233338)
Affinity DataIC50:  6.11E+3nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidine to thymine after 4 to 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439114(CHEMBL2418078)
Affinity DataIC50:  8.54E+3nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192121(2-(4-(1-(4-chlorobenzoyl)-3-(1H-indol-3-yl)-4,5-di...)
Affinity DataIC50:  8.67E+3nMpH: 8.0 T: 2°CAssay Description:The in vitro AChE inhibitory activity was measured using the methods described earlier [Biochem. Pharmacol. 7:88-95]. Briefly, stock solutions (1mg/m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004460(CHEMBL3233327)
Affinity DataIC50:  9.07E+3nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidine to thymine after 4 to 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192117((3-(1H-indol-3-yl)-5-phenyl-4,5-dihydropyrazol-1-y...)
Affinity DataIC50:  9.72E+3nMpH: 8.0 T: 2°CAssay Description:The in vitro AChE inhibitory activity was measured using the methods described earlier [Biochem. Pharmacol. 7:88-95]. Briefly, stock solutions (1mg/m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439115(CHEMBL2418077)
Affinity DataIC50:  9.92E+3nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004468(CHEMBL3233330)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidine to thymine after 4 to 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192114(3-(1H-indol-3-yl)-5-phenyl-4,5-dihydropyrazol-1-yl...)
Affinity DataIC50:  1.06E+4nMpH: 8.0 T: 2°CAssay Description:The in vitro AChE inhibitory activity was measured using the methods described earlier [Biochem. Pharmacol. 7:88-95]. Briefly, stock solutions (1mg/m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439106(CHEMBL2418074)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192122(Ascorbic acid)
Affinity DataIC50:  1.15E+4nMT: 2°CAssay Description:The ABTS free radical cation scavenging ability of the synthe- sized compounds was determined according to the procedure described earlier [Free Radi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004472(CHEMBL3233334)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidine to thymine after 4 to 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192120(2-(4-(1-benzoyl-3-(1H-indol-3-yl)-4,5-dihydro-1H-p...)
Affinity DataIC50:  1.26E+4nMT: 2°CAssay Description:The ABTS free radical cation scavenging ability of the synthe- sized compounds was determined according to the procedure described earlier [Free Radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192122(Ascorbic acid)
Affinity DataIC50:  1.28E+4nMT: 2°CAssay Description:Preparation of DPPH solution was adopted from Molyneux [J. Sci. Technol. 26(2):211-219] and Blois [Nature 181(4617):1199-1200] with minor modificatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439116(CHEMBL2418076)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192116((3-(1H-indol-3-yl)-5-phenyl-4,5-dihydropyrazol-1-y...)
Affinity DataIC50:  1.31E+4nMT: 2°CAssay Description:The ABTS free radical cation scavenging ability of the synthe- sized compounds was determined according to the procedure described earlier [Free Radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192121(2-(4-(1-(4-chlorobenzoyl)-3-(1H-indol-3-yl)-4,5-di...)
Affinity DataIC50:  1.34E+4nMT: 2°CAssay Description:The ABTS free radical cation scavenging ability of the synthe- sized compounds was determined according to the procedure described earlier [Free Radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192116((3-(1H-indol-3-yl)-5-phenyl-4,5-dihydropyrazol-1-y...)
Affinity DataIC50:  1.35E+4nMT: 2°CAssay Description:Preparation of DPPH solution was adopted from Molyneux [J. Sci. Technol. 26(2):211-219] and Blois [Nature 181(4617):1199-1200] with minor modificatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439113(CHEMBL2418079)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192120(2-(4-(1-benzoyl-3-(1H-indol-3-yl)-4,5-dihydro-1H-p...)
Affinity DataIC50:  1.38E+4nMT: 2°CAssay Description:Preparation of DPPH solution was adopted from Molyneux [J. Sci. Technol. 26(2):211-219] and Blois [Nature 181(4617):1199-1200] with minor modificatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004469(CHEMBL3233331)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidine to thymine after 4 to 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192121(2-(4-(1-(4-chlorobenzoyl)-3-(1H-indol-3-yl)-4,5-di...)
Affinity DataIC50:  1.49E+4nMT: 2°CAssay Description:Preparation of DPPH solution was adopted from Molyneux [J. Sci. Technol. 26(2):211-219] and Blois [Nature 181(4617):1199-1200] with minor modificatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192117((3-(1H-indol-3-yl)-5-phenyl-4,5-dihydropyrazol-1-y...)
Affinity DataIC50:  1.54E+4nMT: 2°CAssay Description:Preparation of DPPH solution was adopted from Molyneux [J. Sci. Technol. 26(2):211-219] and Blois [Nature 181(4617):1199-1200] with minor modificatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192117((3-(1H-indol-3-yl)-5-phenyl-4,5-dihydropyrazol-1-y...)
Affinity DataIC50:  1.55E+4nMT: 2°CAssay Description:The ABTS free radical cation scavenging ability of the synthe- sized compounds was determined according to the procedure described earlier [Free Radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192119(2-(4-(1-(2,4-dinitrobenzoyl)-3-(1H-indol-3-yl)-4,5...)
Affinity DataIC50:  1.60E+4nMT: 2°CAssay Description:Preparation of DPPH solution was adopted from Molyneux [J. Sci. Technol. 26(2):211-219] and Blois [Nature 181(4617):1199-1200] with minor modificatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192115((3-(1H-indol-3-yl)-5-phenyl-4,5-dihydropyrazol-1-y...)
Affinity DataIC50:  1.61E+4nMT: 2°CAssay Description:The ABTS free radical cation scavenging ability of the synthe- sized compounds was determined according to the procedure described earlier [Free Radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192119(2-(4-(1-(2,4-dinitrobenzoyl)-3-(1H-indol-3-yl)-4,5...)
Affinity DataIC50:  1.62E+4nMT: 2°CAssay Description:The ABTS free radical cation scavenging ability of the synthe- sized compounds was determined according to the procedure described earlier [Free Radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192115((3-(1H-indol-3-yl)-5-phenyl-4,5-dihydropyrazol-1-y...)
Affinity DataIC50:  1.74E+4nMT: 2°CAssay Description:Preparation of DPPH solution was adopted from Molyneux [J. Sci. Technol. 26(2):211-219] and Blois [Nature 181(4617):1199-1200] with minor modificatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439111(CHEMBL2418057)
Affinity DataIC50:  1.98E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50004471(CHEMBL3233333)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli assessed as conversion of thymidine to thymine after 4 to 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439117(CHEMBL2418075)
Affinity DataIC50:  2.19E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439119(CHEMBL2418072)
Affinity DataIC50:  2.19E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439122(CHEMBL2418069)
Affinity DataIC50:  2.21E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439131(CHEMBL2418085)
Affinity DataIC50:  2.21E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50439112(CHEMBL2418056)
Affinity DataIC50:  2.24E+4nMAssay Description:Inhibition of human recombinant thymidine phosphorylase expressed in Escherichia coli using thymidine as substrate after 4 to 20 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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